Strategies for Enhancing Non-small Cell Lung Cancer Treatment: Integrating Chinese Herbal Medicines with Epidermal Growth Factor Receptor-Tyrosine Kinase …

L Chen, WD Chen, YX Xu, YY Ren, C Zheng… - European Journal of …, 2024 - Elsevier
Non-small cell lung cancer (NSCLC) poses a global health threat, and epidermal growth
factor receptor-tyrosine kinase inhibitors (EGFR-TKIs) such as gefitinib, afatinib, and …

Notch induces transcription by stimulating release of paused RNA polymerase II

JM Rogers, CA Mimoso, BJE Martin… - Genes & …, 2024 - genesdev.cshlp.org
Notch proteins undergo ligand-induced proteolysis to release a nuclear effector that
influences a wide range of cellular processes by regulating transcription. Despite years of …

Temporal dynamics and stoichiometry in human Notch signaling from Notch synaptic complex formation to nuclear entry of the Notch intracellular domain

L Tveriakhina, G Scanavachi, ED Egan… - Developmental Cell, 2024 - cell.com
Mammalian Notch signaling occurs when the binding of Delta or Jagged to Notch stimulates
the proteolytic release of the Notch intracellular domain (NICD), which enters the nucleus to …

Loss of Notch dimerization perturbs intestinal homeostasis by a mechanism involving HDAC activity

Q Dai, K Preusse, D Yu, RA Kovall, K Thorner… - PLoS …, 2024 - journals.plos.org
A tri-protein complex containing NICD, RBPj and MAML1 binds DNA as monomer or as
cooperative dimers to regulate transcription. Mice expressing N otch d imerization-d eficient …

Notch induces transcription by stimulating release of paused RNA Polymerase II

JM Rogers, CA Mimoso, BJE Martin, AP Martin… - bioRxiv, 2024 - biorxiv.org
Notch proteins undergo ligand-induced proteolysis to release a nuclear effector that
influences a wide range of cellular processes by regulating transcription. Despite years of …

Notch Interaction with Glycogen Synthase Kinase-3β in Neurodegenerative Disease

T Traub - 2024 - dspace.cuni.cz
Glycogen synthase kinase-3βeta (GSK-3β) is a serine/threonine protein kinase involved in a
number of signaling processes. Pharmacological inhibition of GSK-3β has been shown to …