The review deals with the pharmaceutically and agrochemically important group of 1, 2, 4-
triazolo [1, 5-a] pyrimidines (TPs) and covers relevant literature published from about 2006 …

[1, 2, 4] Triazolo [1, 5-a] pyrimidines are very interesting and trend class of fused
heterocycles due to their valuable biological properties. Some [1, 2, 4]-triazolo [1, 5-a] …

β-Ketothioamides (KTAs) are versatile building blocks for the rapid construction of various
heterocyclic compounds. In the past decade, a number of successful reactions based on …

1, 2, 4-Triazole moieties have been incorporated into a wide variety of therapeutically
interesting drug candidates including central nervous system stimulants, sedatives …

A mild and straightforward synthetic protocol for construction of a furan skeleton promoted by
Yb (OTf) 3 from β-ketothioamides and arylglyoxals has been developed at room …

A diversity of new 7‐substituted [1, 2, 4] triazolo [1, 5‐a] pyrimidine and 6‐substituted [1, 2, 4]
triazolo [1, 5‐a] pyrimidine‐7‐amine derivatives has been synthesized via reaction of 3 …

摘要建立了一种以β-芳甲酰硫代酰胺(KTAs) 和丙二腈为合成砌块合成噻唑啉衍生物的新方法.
采用廉价的四正丁基碘化胺(TBAI)/叔丁基过氧化氢(TBHP) 为催化氧化体系, 在三乙胺存在下 …

β-Ketothioamides (KTAs) have proved to be important precursors to furnish diverse
heterocyclic moieties over the last couple of decades. The convergence of reactive sites and …

Two novel N-heterocyclic carbene-palladium (II) complexes were conveniently synthesized
through one-pot reactions of imidazolium salts, palladium chloride and acridine. The new …