Recent approaches to the synthesis of tetrahydrocarbazoles
TY Chaudhari, V Tandon - Organic & Biomolecular Chemistry, 2021 - pubs.rsc.org
The tetrahydrocarbazole (THC) motif is ubiquitous in natural products and biologically active
compounds. THCs can serve as favorable synthetic intermediates or precursors en-route to …
compounds. THCs can serve as favorable synthetic intermediates or precursors en-route to …
2-Phenylbenzofuran derivatives as butyrylcholinesterase inhibitors: synthesis, biological activity and molecular modeling
A series of 2-phenylbenzofurans compounds was designed, synthesized and evaluated as
cholinesterase inhibitors. The biological assay experiments showed that most of the …
cholinesterase inhibitors. The biological assay experiments showed that most of the …
Synthesis and molecular docking studies of some 4-phthalimidobenzenesulfonamide derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors
A series of 4-phthalimidobenzenesulfonamide derivatives were designed, synthesized and
evaluated for the inhibitory activities against acetylcholinesterase (AChE) and …
evaluated for the inhibitory activities against acetylcholinesterase (AChE) and …
N-Alkylated 1,4-Diazabicyclo[2.2.2]octane–Polyethylene Glycol Melt as Deep Eutectic Solvent for the Synthesis of Fisher Indoles and 1H-Tetrazoles
1, 4-Diazabicyclo [2.2. 2] octane (DABCO)-based ionic liquids (ILs) 2–4 were synthesized by
the N-alkylation of DABCO using alkyl halides of varying chain lengths (C2, C5, and C7) …
the N-alkylation of DABCO using alkyl halides of varying chain lengths (C2, C5, and C7) …
Microwave-assisted organic synthesis, structure–activity relationship, kinetics and molecular docking studies of non-cytotoxic benzamide derivatives as selective …
A series of benzamide derivatives 1–12 with various functional groups (–H,–Br,–F,–OCH 3,–
OC 2 H 5, and–NO 2) was synthesized using an economic, and facile Microwave-Assisted …
OC 2 H 5, and–NO 2) was synthesized using an economic, and facile Microwave-Assisted …
Engaging Diastereomeric syn‐ and anti‐6‐Bromo‐4a‐isopropyl‐2‐methyl‐2,3,4,4a‐tetrahydro‐1H‐carbazoles in Suzuki Coupling Reaction: Synthesis, Spectral …
Suzuki coupling reaction is one of the useful methods for carbon‐carbon bond formation. In
the present study, the aforementioned method is used to expand an aryl appendage on the …
the present study, the aforementioned method is used to expand an aryl appendage on the …
Isolation, Derivatization, in-vitro, and in-silico Studies of Potent Butyrylcholinesterase Inhibitors from Berberis parkeriana Schneid
Seven known isoquinoline alkaloids 1–7 were isolated from the root extracts of Berberis
parkeriana Schneid. Nine new derivatives 8–16 of one of the isolated compounds …
parkeriana Schneid. Nine new derivatives 8–16 of one of the isolated compounds …
Fischer indolization of terpenes and steroids
S Kotha, P Meher - ChemistrySelect, 2024 - Wiley Online Library
Here we report a new synthetic approach to several intricate indoles and hydrazones
starting with commercially available terpenes and steroids via Fischer indolization (FI) …
starting with commercially available terpenes and steroids via Fischer indolization (FI) …
Synthesis, biological evaluation, and docking studies of some 5‐chloro‐2(3H)‐benzoxazolone Mannich bases derivatives as cholinesterase inhibitors
A series of N‐substituted‐5‐chloro‐2 (3H)‐benzoxazolone derivatives were synthesized
and evaluated for their acetylcholinesterase (AChE), butyrylcholinesterase (BuChE) …
and evaluated for their acetylcholinesterase (AChE), butyrylcholinesterase (BuChE) …
[PDF][PDF] Exploring the diastereoselectivity for Fischer indolization of L-menthone under different conditions, spectral characterization, and biological activities of new (2R …
S Rasheed, R Sadiq, FZ Basha - European Journal of Chemistry, 2022 - academia.edu
Tetrahydrocarbazole is defined as an indole skeleton fused with a cyclohexane ring. This
class is widely distributed in nature and has gained immense attention of medicinal chemists …
class is widely distributed in nature and has gained immense attention of medicinal chemists …