Review on the diverse biological effects of glabridin

J Zhang, X Wu, B Zhong, Q Liao, X Wang… - Drug Design …, 2023 - Taylor & Francis
Glabridin is a prenylated isoflavan from the roots of Glycyrrhiza glabra Linne and has posed
great impact on the areas of drug development and medicine, due to various biological …

Glabridin ameliorates methotrexate-induced liver injury via attenuation of oxidative stress, inflammation, and apoptosis

A Dogra, D Gupta, S Bag, I Ahmed, S Bhatt, E Nehra… - Life Sciences, 2021 - Elsevier
Despite unprecedented advances in modern medicine, no safe and effective drug is
available to date for oral administration to combat drug-induced liver injury, which is a vital …

Isolation and anticancer activity evaluation of rare Bisaryl anthraquinone antibiotics from novel Streptomyces sp. strain of NW Himalayan region

RS Manhas, SM Ahmad, KB Mir, A Ahmed… - Chemico-Biological …, 2022 - Elsevier
Biosynthesis of bisaryl preanthraquinone antibiotics by various microorganisms differs in
monomeric subunits as well as their dimerization positions leading to different …

Molecular mechanism for the involvement of CYP2E1/NF-κB axis in bedaquiline-induced hepatotoxicity

P Kotwal, P Khajuria, S Dhiman, D Kour, SK Dhiman… - Life Sciences, 2023 - Elsevier
Bedaquiline (BDQ) is a new class of anti-tubercular (anti-TB) drugs and is currently reserved
for multiple drug resistance (MDR-TB). However, after receiving fast-track approval, its …

Effect of Myricetin on CYP2C8 Inhibition to Assess the Likelihood of Drug Interaction Using In Silico, In Vitro, and In Vivo Approaches

S Bhatt, D Manhas, V Kumar, A Gour, K Sharma… - ACS …, 2022 - ACS Publications
Myricetin, a bioflavonoid, is widely used as functional food/complementary medicine and
has promising multifaceted pharmacological actions against therapeutically validated …

Rottlerin renders a selective and highly potent CYP2C8 inhibition to impede EET formation for implication in cancer therapy

D Manhas, S Bhatt, G Rai, V Kumar, S Bharti… - Chemico-biological …, 2023 - Elsevier
CYP2C8 is a crucial CYP isoform responsible for the metabolism of xenobiotics and
endogenous molecules. CYP2C8 converts arachidonic acid to epoxyeicosatrienoic acids …

Glabridin attenuates paracetamol-induced liver injury in mice via CYP2E1-mediated inhibition of oxidative stress

S Bhatt, A Sharma, A Dogra, P Sharma… - Drug and Chemical …, 2022 - Taylor & Francis
CYP2E1 plays a crucial role in the bio-activation of toxic substances leading to liver
damage. In this context, CYP2E1 converts paracetamol (PCM) to N-acetyl-p-benzoquinone …

Identification of Cytochrome P450 2E1 as a Novel Target in Glioma and Development of Its Inhibitor as an Anti‐Tumor Agent

G Hu, Y Fang, H Xu, G Wang, R Yang, F Gao… - Advanced …, 2023 - Wiley Online Library
Glioblastoma (GBM) is a devastating inflammation‐related cancer for which novel
therapeutic targets are urgently required. Previous studies of the authors indicate …

Development of mupirocin-impregnated bacterial cellulosic transdermal patches for the management of skin infection

R Bhat, A Dogra, S Chib, M Kumar, IA Khan… - ACS …, 2024 - ACS Publications
The present study reports the production of bacterial cellulose (BC) membranes using
Komagataeibacter hansenii for the development of transdermal wound healing patches. BC …

Glabridin plays dual action to intensify anti-metastatic potential of paclitaxel via impeding CYP2C8 in liver and CYP2J2/EETs in tumor of an orthotopic mouse model of …

A Jamwal, J Chand, A Dash, S Bhatt, S Dhiman… - Chemico-Biological …, 2023 - Elsevier
In spite of unprecedented advances in modern cancer therapy, there is still a dearth of
targeted therapy to circumvent triple-negative breast cancer (TNBC). Paclitaxel is the front …