Investigating 1, 2, 3, 4, 5, 6-hexahydroazepino [4, 3-b] indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for …

R Purgatorio, M de Candia, M Catto, A Carrieri… - European Journal of …, 2019 - Elsevier
Due to the role of butyrylcholinesterase (BChE) in acetylcholine hydrolysis in the late stages
of the Alzheimer's disease (AD), inhibitors of butyrylcholinesterase (BChE) have been …

A new approach to construction of isoindolo [1, 2-a] isoquinoline alkaloids Nuevamine, Jamtine, and Hirsutine via IMDAF reaction

FI Zubkov, JD Ershova, AA Orlova, VP Zaytsev… - Tetrahedron, 2009 - Elsevier
The interaction between 1-furyl-1, 2, 3, 4-tetrahydroisoquinolines and unsaturated acids
derivatives (acryloyl, methacryloyl, and crotonoyl chloride, maleic and citraconic anhydride) …

Ester derivatives of annulated tetrahydroazocines: A new class of selective acetylcholinesterase inhibitors

A Carotti, M de Candia, M Catto, TN Borisova… - Bioorganic & medicinal …, 2006 - Elsevier
A series of ester derivatives of annulated tetrahydroazocines, namely 2, 3, 6, 11-tetrahydro-
1H-azocino [4, 5-b] indoles (5–10), 2, 3, 6, 7-tetrahydro-1H-azocino [5, 4-b] indoles (11–14) …

A concise approach toward tetrazolyl-substituted benzazocines via a novel isocyanide-based multicomponent reaction

RS Borisov, LG Voskressensky, AI Polyakov… - Synlett, 2014 - thieme-connect.com
The synthesis of pharmacologically relevant isoquinoline-tetrazoles and benzazocine-
tetrazoles via sequential azido-Ugi and alkyne-induced ring-expansion reactions starting …

The interaction of 4-hydroxymethyl isoindolines with dehydrobenzene. Synthesis of 3-phenylaminomethyldihydrobenzo [c] furanes

AV Varlamov, NI Guranova, TN Borisova, FAA Toze… - Tetrahedron, 2015 - Elsevier
The interaction of 4-hydroxymethyl isoindolines with dehydrobenzene. Synthesis of 3-phenylaminomethyldihydrobenzo[c]furanes
- ScienceDirect Skip to main contentSkip to article Elsevier logo Journals & Books Search …

Tetrahydropyridine (THP) ring expansion under the action of activated terminal alkynes. The first synthesis and X-ray crystal structure of tetrahydropyrimido [4, 5-d] …

LG Voskressensky, TN Borisova, IS Kostenev… - Tetrahedron letters, 2006 - Elsevier
Tetrahydropyridopyrimidines (THPPm) underwent tandem cleavage–cyclization piperidine
ring enlargement under the action of terminal activated alkynes to produce …

Transformations of tetrahydro-pyrido[4,3-d]pyrimidines [b]-condensed with isoxazole, thiazole, thiadiazole, and triazole units under the action of activated alkynes

LG Voskressensky, TN Borisova, MV Ovcharov… - Chemistry of …, 2008 - Springer
It has been established that 5-vinyl-substituted (NR, N-vinylaminomethyl) isoxazolo
(thiazolo, thiadiazolo) pyrimidines are formed when tetrahydropyrido [3, 4-d] pyrimidines …

Reaction of 1-substituted tetrahydro-β-carbolines with activated alkynes-a new original approach to the synthesis of tetrahydroazocino[5,4-b]indoles

LG Voskressensky, TN Borisova, LN Kulikova… - Chemistry of …, 2007 - Springer
The transformations of 1-substituted tetrahydro-β-carbolines by the action of activated
alkynes were studied. The action of dimethyl acetylenedicarboxylate in methanol gives …

γ-Carbolines and their hydrogenated derivatives 3.* Hydrogenated derivatives of γ-carbolines: chemical and biological poperties

RS Alekseyev, AV Kurkin, MA Yurovskaya - Chemistry of heterocyclic …, 2011 - Springer
γ-Carbolines and their hydrogenated derivatives 3.* Hydrogenated derivatives of γ-carbolines:
chemical and biological poperties (Review) | Chemistry of Heterocyclic Compounds Skip to …

Recyclization of benzofuropyridines by the action of activated alkynes in the synthesis of spiro [benzofuropyridines], representatives of a new class of …

LG Voskressensky, SA Kovaleva, TN Borisova… - Chemistry of …, 2013 - Springer
A study was carried out on the domino transformations of tetrahydrobenzofuro [2, 3-c]
pyridines and tetrahydrobenzofuro [3, 2-c] pyridines by the action of activated alkynes in …