Recent developments in azole compounds as antibacterial and antifungal agents
XM Peng, GX Cai, CH Zhou - Current Topics in Medicinal …, 2013 - ingentaconnect.com
Azole compounds are an important class of nitrogen heterocycles with electron-rich
property. This special structure endows azole-based derivatives easily bind with the …
property. This special structure endows azole-based derivatives easily bind with the …
[HTML][HTML] Synthesis and inhibition profiles of N-benzyl-and N-allyl aniline derivatives against carbonic anhydrase and acetylcholinesterase–A molecular docking study
The alkyl and aryl derivatives of aniline are important starting materials in fine organic
synthesis. Allyl bromide and benzyl chloride were taken as substrates for the alkylation …
synthesis. Allyl bromide and benzyl chloride were taken as substrates for the alkylation …
Investigation of inhibitory properties of some hydrazone compounds on hCA I, hCA II and AChE enzymes
Recently, inhibition of carbonic anhydrase (hCA) and acetylcholinesterase (AChE) have
appeared as a promising approach for pharmacological intervention in a variety of disorders …
appeared as a promising approach for pharmacological intervention in a variety of disorders …
Antimicrobial activity and a SAR study of some novel benzimidazole derivatives bearing hydrazone moiety
In this study 12 novel benzimidazole compounds bearing hydrazone moiety were
synthesized in order to investigate their possible antibacterial and antifungal activity …
synthesized in order to investigate their possible antibacterial and antifungal activity …
Efficient synthesis, antibacterial, antifungal, antioxidant and cytotoxicity study of 2‐(2‐hydrazineyl) thiazole derivatives
VA Adole, RA More, BS Jagdale, TB Pawar… - …, 2020 - Wiley Online Library
In the present investigation, an alluring green PEG‐400 mediated one‐pot synthesis of
novel 2‐(2‐hydrazinyl) thiazole derivatives from 1, 2, 6, 7‐tetrahydro‐8H‐indeno [5, 4‐b] …
novel 2‐(2‐hydrazinyl) thiazole derivatives from 1, 2, 6, 7‐tetrahydro‐8H‐indeno [5, 4‐b] …
[PDF][PDF] Therapeutic review exploring antimicrobial potential of hydrazones as promising lead
G Uppal, S Bala, S Kamboj, M Saini - Der Pharma Chemica, 2011 - researchgate.net
This review includes detailed study of structures of various hydrazones synthesized and
evaluated for their antimicrobial activity. Hydrazone is a class of organic compounds with …
evaluated for their antimicrobial activity. Hydrazone is a class of organic compounds with …
Design, synthesis and mode of action of some benzothiazole derivatives bearing an amide moiety as antibacterial agents
In this study ten benzothiazole derivatives bearing the amide moiety were designed,
synthesized and evaluated for their antibacterial activity and possible mode of action …
synthesized and evaluated for their antibacterial activity and possible mode of action …
Design, Synthesis, and Pharmacological Evaluation of N-Acylhydrazones and Novel Conformationally Constrained Compounds as Selective and Potent Orally Active …
AE Kümmerle, M Schmitt, SVS Cardozo… - Journal of medicinal …, 2012 - ACS Publications
Among a small series of tested N-acylhydrazones (NAHs), the compound 8a was selected
as a selective submicromolar phosphodiesterase-4 (PDE4) inhibitor associated with anti …
as a selective submicromolar phosphodiesterase-4 (PDE4) inhibitor associated with anti …
Synthesis of some new [1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazines and [1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazoles starting from 5-nitro-2-furoic acid and evaluation of …
SMI Badr, RM Barwa - Bioorganic & medicinal chemistry, 2011 - Elsevier
New series of fused 1, 2, 4-triazoles such as, 6-(aryl)-3-(5-nitrofuran-2-yl)-5, 6-dihydro-[1, 2,
4] triazolo [3, 4-b][1, 3, 4] thiadiazoles 4–8, 6-(alkyl/aryl amino)-3-(5-nitrofuran-2-yl)-[1, 2, 4] …
4] triazolo [3, 4-b][1, 3, 4] thiadiazoles 4–8, 6-(alkyl/aryl amino)-3-(5-nitrofuran-2-yl)-[1, 2, 4] …
Synthesis, structural and spectroscopic features, and investigation of bioactive nature of a novel organic-inorganic hybrid material 1H-1, 2, 4-triazole-4-ium …
The novel inorganic-organic hybrid material 1H-1, 2, 4-triazole-4-ium trioxonitrate (TAN)
have been elaborated and crystallized to the monoclinic system with space group P2 1/c …
have been elaborated and crystallized to the monoclinic system with space group P2 1/c …