A key review on oxadiazole analogs as potential methicillin-resistant Staphylococcus aureus (MRSA) activity: Structure-activity relationship studies
Methicillin-resistant Staphylococcus aureus (MRSA) is becoming dangerous to human
beings due to easy transmission mode and leading to the difficult-to-treat situation. The rapid …
beings due to easy transmission mode and leading to the difficult-to-treat situation. The rapid …
The antibacterial activity of 1, 2, 3-triazole-and 1, 2, 4-triazole-containing hybrids against Staphylococcus aureus: An updated review (2020-present)
J Li, J Zhang - Current Topics in Medicinal Chemistry, 2022 - ingentaconnect.com
Staphylococcus aureus (S. aureus), a prominent, highly contagious nosocomial and
community-acquired bacterial pathogen, can cause a broad spectrum of diseases. Antibiotic …
community-acquired bacterial pathogen, can cause a broad spectrum of diseases. Antibiotic …
Fluorinated azoles as effective weapons in fight against methicillin-resistance staphylococcus aureus (MRSA) and its SAR studies
The rapid spread of Methicillin-resistant Staphylococcus aureus (MRSA) and its difficult-to-
treat skin and filmsy diseases are making MRSA a threat to human life. The most dangerous …
treat skin and filmsy diseases are making MRSA a threat to human life. The most dangerous …
Identification of 1, 3, 4-oxadiazoles as tubulin-targeted anticancer agents: a combined field-based 3D-QSAR, pharmacophore model-based virtual screening …
Cancer is one of the most prominent causes of death worldwide and tubulin is a crucial
protein of cytoskeleton that maintains essential cellular functions including cell division as …
protein of cytoskeleton that maintains essential cellular functions including cell division as …
Thiophene‐containing compounds with antimicrobial activity
G Roman - Archiv der Pharmazie, 2022 - Wiley Online Library
Thiophene, as a member of the group of five‐membered heterocycles containing one
heteroatom, is one of the simplest heterocyclic systems. Many synthetic strategies allow the …
heteroatom, is one of the simplest heterocyclic systems. Many synthetic strategies allow the …
Synthesis, intramolecular cyclization, and antinociceptive activity of 4-(het) aryl-2-{[4-(4-chlorophenyl)-3-(ethoxycarbonyl) thiophen-2-yl] amino}-4-oxobut-2-enoic …
Synthesis and intramolecular cyclization of the substituted 4-(het) aryl-2-{[4-(4-chlorophenyl)-
3-(ethoxycarbonyl) thiophen-2-yl] amino}-4-oxobut-2-enoic acids were studied. It was found …
3-(ethoxycarbonyl) thiophen-2-yl] amino}-4-oxobut-2-enoic acids were studied. It was found …
Quinazoline clubbed thiazole and 1, 3, 4-oxadiazole heterocycles: synthesis, characterization, antibacterial evaluation, and molecular docking studies
In search of potent antibacterial agents, a series of novel quinazolines, bearing thiazole and
1, 3, 4-oxadiazole heterocycles 6a–j (3-(4-methyl-5-(4-((arylamino) methyl)-5-thioxo-4, 5 …
1, 3, 4-oxadiazole heterocycles 6a–j (3-(4-methyl-5-(4-((arylamino) methyl)-5-thioxo-4, 5 …
An effective green one-pot synthesis of some novel 5-(thiophene-2-carbonyl)-6-(trifluoromethyl)pyrano[2,3-c]pyrazoles and 6-(thiophene-2-carbonyl)-7-(trifluoromethyl)pyrano[2 …
An effective green one-pot and catalyst-free synthesis of a series of novel 5-(thiophene-2-
carbonyl)-6-(trifluoromethyl) pyrano [2, 3-c] pyrazoles and 6-(thiophene-2-carbonyl)-7 …
carbonyl)-6-(trifluoromethyl) pyrano [2, 3-c] pyrazoles and 6-(thiophene-2-carbonyl)-7 …
Linear and Branched Forms of Short Antimicrobial Peptide-IRK Inhibit Growth of Multi Drug Resistant Staphylococcus aureus Isolates from Mastitic Cow Milk
Antimicrobial peptides (AMPs) offer a novel alternative to present day antibiotics which are
becoming ineffective due to development of resistance in microbes. In this study, a short …
becoming ineffective due to development of resistance in microbes. In this study, a short …
One-Pot Three-Component Synthesis of a Series of 2-Amino-4-(4-oxo-4H-chromen-3-yl)-5-(2,2,2-trifluoroacetyl)-6-(trifluoromethyl)-4H-pyrans and 2-Amino-4-(4-oxo-4H …
TE Ali, MA Assiri, AA Shati, MY Alfaifi… - Russian Journal of …, 2022 - Springer
Abstract Novel functionalized 2-amino-4-(4-oxo-4 H-chromen-3-yl)-5-(2, 2, 2-trifluoroacetyl)-
6-(trifluoromethyl)-4 H-pyrans and 2-amino-4-(4-oxo-4 H-chromen-3-yl)-5-(thiophene-2 …
6-(trifluoromethyl)-4 H-pyrans and 2-amino-4-(4-oxo-4 H-chromen-3-yl)-5-(thiophene-2 …