Cinnamic acid and its phenolic analogues are natural substances. Chemically, cinnamic
acids or the 3-phenyl acrylic acids, offer three main reactive sites: substitution on the phenyl …

Abstract A novel series of 1, 4-naphthoquinones (33–44) tethered by open and closed chain
sulfonamide moieties were designed, synthesized and evaluated for their cytotoxic and …

Abstract p‐Nitrobenzyloxycarbonyl (pNZ) was used as a temporary protecting group for α‐
amino functionalities in solid‐phase peptide synthesis. The corresponding derivatives are …

We have described compound 1 as a lead structure for a novel class of anti-malarial agents.
Replacement of the 3-phenylpropionyl moiety of the lead structure 1 by a 4-propoxycinnamic …

[(p-Cymene) Ru (2, 2′-bpyO)(H2O)] was proven to be an efficient catalyst for the synthesis
of amino-(N-alkyl) benzenesulfonamides via selective N-alkylation of …

Aldose reductase (ALR2) is a crucial enzyme in the development of the major complications
of diabetes mellitus. Very recently it has been demonstrated that the ARL2 inhibitor …

The creation of caged molecules involves the attachment of protecting groups to biologically
active compounds such as ligands, substrates and drugs that can be removed under specific …

R, is an alkyl residue containing 6 to 20 carbon atoms, or an alkene residue containing from
9 to 25 carbon atoms with 1 to 6 double bonds, R, together with the carbonyl group to which …

Background: Now a day's green synthesis for multicomponent reactions is a powerful tool for
construction of five membered/six membered heterocyclic ring systems. The synthesis of …

US10856563B2 - N-acyl-amino acid derivatives for improvement of the flavor profile of edible
compositions - Google Patents US10856563B2 - N-acyl-amino acid derivatives for improvement …