Catalytic functionalization of indoles in a new dimension
M Bandini, A Eichholzer - Angewandte Chemie International …, 2009 - Wiley Online Library
Abstract 140 Years ago Adolf von Baeyer proposed the structure of a heteroaromatic
compound which revolutionized organic and medical chemistry: indole. After more than a …
compound which revolutionized organic and medical chemistry: indole. After more than a …
Bis-and trisindolylmethanes (BIMs and TIMs)
The indole ring system is present in many natural products, pharmaceuticals,
agrochemicals, and other compounds of importance. 1–8 The indole unit forms the basis for …
agrochemicals, and other compounds of importance. 1–8 The indole unit forms the basis for …
Synthetic approaches to 3-(2-nitroalkyl) indoles and their use to access tryptamines and related bioactive compounds
S Lancianesi, A Palmieri, M Petrini - Chemical Reviews, 2014 - ACS Publications
The assembly of architecturally complex alkaloids embedding the indole nucleus is of
paramount importance for the target oriented synthesis of biologically active molecules. 1 A …
paramount importance for the target oriented synthesis of biologically active molecules. 1 A …
Katalytische Funktionalisierung von Indolen in einer neuen Dimension
M Bandini, A Eichholzer - Angewandte Chemie, 2009 - Wiley Online Library
Abstract Vor 140 Jahren schlug Adolf von Baeyer die Struktur für eine heteroaromatische
Verbindung vor, die die organische und medizinische Chemie nachhaltig veränderte: Indol …
Verbindung vor, die die organische und medizinische Chemie nachhaltig veränderte: Indol …
Functionalization of indole and pyrrole cores via Michael-type additions
N Saracoglu - Bioactive Heterocycles V, 2007 - Springer
The Michael reaction has been the subject of numerous reviews. Furthermore, the first
review on anti-Michael addition has been published. The present review focuses only on the …
review on anti-Michael addition has been published. The present review focuses only on the …
Recent Developments in the Synthesis of Indole‐Pyrazole Hybrids
Indole and pyrazole are two important scaffolds in the field of medicinal chemistry.
Compounds bearing indole and/or pyrazole moiety have been extensively investigated for a …
Compounds bearing indole and/or pyrazole moiety have been extensively investigated for a …
2-Aminopyridinium ions activate nitroalkenes through hydrogen bonding
N Takenaka, RS Sarangthem, SK Seerla - Organic Letters, 2007 - ACS Publications
2-Aminopyridinium ions were found to activate nitroalkenes toward conjugate addition of
heteroaromatic compounds with low catalyst loadings and the Diels− Alder reaction with the …
heteroaromatic compounds with low catalyst loadings and the Diels− Alder reaction with the …
Synthesis of bis (indolyl) alkanes by a site-selective gold-catalyzed addition of indoles to butynol derivatives
J Barluenga, A Fernández, F Rodríguez… - Journal of Organometallic …, 2009 - Elsevier
A new site-selective hydroarylation reaction of alkynes catalyzed by gold complexes and
directed by an internal hydroxyl group has been developed. Thus, the treatment of 3-butyn-1 …
directed by an internal hydroxyl group has been developed. Thus, the treatment of 3-butyn-1 …
[PDF][PDF] Heteoropoly Acids: Green Chemical Catalysts in Organic Synthesis
T Ueda, H Kotsuki - Heterocycles, 2008 - triggered.edina.clockss.org
Heteropoly acids have been used in various fields of organic synthesis mainly due to their
characteristic features: they are cost-effective reagents that are strongly acidic …
characteristic features: they are cost-effective reagents that are strongly acidic …
Ce III-promoted oxidation. Efficient aerobic one-pot eco-friendly synthesis of oxidized bis (indol-3-yl) methanes and cyclic tetra (indolyl) dimethanes
Indoles and benzaldehyde derivatives undergo an efficient one-pot smooth condensation
and a further atmospheric-pressure aerobic dehydrogenation with CeCl3 in i-PrOH, to afford …
and a further atmospheric-pressure aerobic dehydrogenation with CeCl3 in i-PrOH, to afford …