Quinoline-based antimalarial hybrid compounds
S Vandekerckhove, M D'hooghe - Bioorganic & medicinal chemistry, 2015 - Elsevier
Quinoline-containing compounds, such as quinine and chloroquine, have a long-standing
history as potent antimalarial agents. However, the increasing resistance of the Plasmodium …
history as potent antimalarial agents. However, the increasing resistance of the Plasmodium …
Rhodanine as a privileged scaffold in drug discovery
Rhodanines, thiazolidine-2, 4-diones and pseudothiohydantoins have become a very
interesting class of heterocyclic compounds since the introduction of various glitazones and …
interesting class of heterocyclic compounds since the introduction of various glitazones and …
Simultaneous improvement of antimicrobial, antifouling, and transport properties of forward osmosis membranes with immobilized highly-compatible polyrhodanine …
A Rahimpour, SF Seyedpour… - … science & technology, 2018 - ACS Publications
This work shows that incorporating highly compatible polyrhodanine nanoparticles (PRh-
NPs) into a polyamide (PA) active layer allows for fabricating forward osmosis (FO) thin-film …
NPs) into a polyamide (PA) active layer allows for fabricating forward osmosis (FO) thin-film …
Thermal properties, antimicrobial activity and DNA binding of Ni (II) complexes of azo dye compounds
A novel series of nickel (II) azo dye complexes of 5-(4-methoxyphenylazo)-2-thioxo-4-
thiazolidinone (HL 1), 5-(4-methylphenylazo)-2-thioxo-4-thiazolidinone (HL 2), 5 …
thiazolidinone (HL 1), 5-(4-methylphenylazo)-2-thioxo-4-thiazolidinone (HL 2), 5 …
Polymer complexes. LXXI. Spectroscopic studies, thermal properties, DNA binding and antimicrobial activity of polymer complexes
Polymer complexes of Co (II), Ni (II), Mn (II), Cr (III) and Cd (II) were prepared by the reaction
of 3‐allyl‐5‐[(4‐nitrophenylazo)]‐2‐thioxothiazolidine‐4‐one (HL) with metal ions. The …
of 3‐allyl‐5‐[(4‐nitrophenylazo)]‐2‐thioxothiazolidine‐4‐one (HL) with metal ions. The …
Drug screening of rhodanine derivatives for antibacterial activity
S Maddila, S Gorle… - Expert Opinion on Drug …, 2020 - Taylor & Francis
Introduction: Bacteriological infections are a major risk to human health. These include all
hospital and public-acquired infections. In drug discovery, rhodanines are privileged …
hospital and public-acquired infections. In drug discovery, rhodanines are privileged …
Synthesis and evaluation of some new fluorinated hydroquinazoline derivatives as antifungal agents
MM Ghorab, SM Abdel-Gawad, MSA El-Gaby - Il Farmaco, 2000 - Elsevier
The key intermediate octahydroquinazoline (1) was obtained in one pot synthesis by a
modification of the Biginelli reaction. Compound 1 was allowed to react with phenacyl …
modification of the Biginelli reaction. Compound 1 was allowed to react with phenacyl …
Synthesis, molecular geometry, spectroscopic studies and thermal properties of Co (II) complexes
Co (II) complexes (1‐4) were prepared and characterized by elemental analyses, infrared
spectra, spectral studies, magnetic susceptibility measurements, X‐ray diffraction analysis …
spectra, spectral studies, magnetic susceptibility measurements, X‐ray diffraction analysis …
Synthesis, spectroscopic, thermal properties, Calf thymus DNA binding and quantum chemical studies of M (II) complexes
A new series of transition metal complexes of Cu (II), Co (II), Ni (II), Mn (II) and Cd (II) were
prepared from the ligand of 5‐(4‐benzenesulfonic acid azo)‐2‐thioxo‐4‐thiazolidinone …
prepared from the ligand of 5‐(4‐benzenesulfonic acid azo)‐2‐thioxo‐4‐thiazolidinone …
Influence of substituent effects on spectroscopic properties and antimicrobial activity of 5-(4′-substituted phenylazo)-2-thioxothiazolidinone derivatives
Abstract 5-(4′-substituted phenylazo)-2-thioxothiazolidinone derivatives (HL n) have been
synthesized and characterized by elemental analysis, spectra (IR, electronic and 1 H NMR) …
synthesized and characterized by elemental analysis, spectra (IR, electronic and 1 H NMR) …