DYRK1A: a down syndrome-related dual protein kinase with a versatile role in tumorigenesis

AJ Laham, M Saber-Ayad, R El-Awady - Cellular and Molecular Life …, 2021 - Springer
Dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) is a dual kinase
that can phosphorylate its own activation loop on tyrosine residue and phosphorylate its …

Doxorubicin-loaded iron oxide nanoparticles for glioblastoma therapy: A combinational approach for enhanced delivery of nanoparticles

M Norouzi, V Yathindranath, JA Thliveris, BM Kopec… - Scientific reports, 2020 - nature.com
Although doxorubicin (DOX) is an effective anti-cancer drug with cytotoxicity in a variety of
different tumors, its effectiveness in treating glioblastoma multiforme (GBM) is constrained by …

A review on the assessment of imidazo [1, 2-a] pyridines as corrosion inhibitor of metals

R Salim, E Ech-Chihbi, H Oudda, F El Hajjaji… - Journal of Bio-and Tribo …, 2019 - Springer
Abstract Imidazo [1, 2-a] pyridines find great importance in several commercially available
drugs but recently, this derivative has been reported as effective corrosion inhibitors due to …

Molecular characterization of the grape seeds extract's effect against chemically induced liver cancer: In vivo and in vitro analyses

AA Hamza, GH Heeba, HM Elwy, C Murali… - Scientific reports, 2018 - nature.com
The purpose of this study was to investigate the anti-cancer property of grape seed extract
(GSE) during early stages of developing liver cancer using a two-stage carcinogenic model …

Enhanced drug delivery using sonoactivatable liposomes with membrane-embedded porphyrins

X Wang, F Yan, X Liu, P Wang, S Shao, Y Sun… - Journal of controlled …, 2018 - Elsevier
Small molecules that interfere with nucleic acid are widely used in chemotherapy, however,
improved delivery approaches are required to improve anti-tumor outcomes. Here, we …

Upregulation of Akt/NF-κB-regulated inflammation and Akt/Bad-related apoptosis signaling pathway involved in hepatic carcinoma process: suppression by carnosic …

B Tang, F Tang, Z Wang, G Qi, X Liang… - International Journal …, 2016 - Taylor & Francis
Primary liver cancer is globally the sixth most frequent cancer, and the second leading
cause of cancer death and its incidence is increasing in many countries, becoming a serious …

Monitoring doxorubicin cellular uptake and trafficking using in vitro Raman microspectroscopy: short and long time exposure effects on lung cancer cell lines

Z Farhane, F Bonnier, HJ Byrne - Analytical and bioanalytical chemistry, 2017 - Springer
Raman microspectroscopy is a non-invasive, in vitro analytical tool which is being
increasingly explored for its potential in clinical applications and monitoring the uptake …

Selenylated Imidazo[1,2-a]pyridine Induces Cell Senescence and Oxidative Stress in Chronic Myeloid Leukemia Cells

GT Burkner, DA Dias, KFS Souza, AJP Araújo… - Molecules, 2023 - mdpi.com
Imidazo [1, 2-a] pyridines (IPs) have been studied regarding drug development. The
objective of this work was to evaluate the antileukemic capacity of IP derivatives by …

Doxorubicin kinetics and effects on lung cancer cell lines using in vitro Raman micro‐spectroscopy: binding signatures, drug resistance and DNA repair

Z Farhane, F Bonnier, O Howe, A Casey… - Journal of …, 2018 - Wiley Online Library
Raman micro‐spectroscopy is a non‐invasive analytical tool, whose potential in cellular
analysis and monitoring drug mechanisms of action has already been demonstrated, and …

Novel selenylated imidazo [1, 2-a] pyridines for breast cancer chemotherapy: Inhibition of cell proliferation by Akt-mediated regulation, DNA cleavage and apoptosis

GM Almeida, J Rafique, S Saba, T Siminski… - Biochemical and …, 2018 - Elsevier
A novel series of selenylated imidazo [1, 2-a] pyridines were designed and synthesized with
a view to a promising activity against breast cancer cell. The compounds, 7-methyl-3 …