[HTML][HTML] Natural products in drug discovery: advances and opportunities

AG Atanasov, SB Zotchev, VM Dirsch… - Nature reviews Drug …, 2021 - nature.com
Natural products and their structural analogues have historically made a major contribution
to pharmacotherapy, especially for cancer and infectious diseases. Nevertheless, natural …

Artificial intelligence for natural product drug discovery

MW Mullowney, KR Duncan, SS Elsayed… - Nature Reviews Drug …, 2023 - nature.com
Developments in computational omics technologies have provided new means to access
the hidden diversity of natural products, unearthing new potential for drug discovery. In …

Systematic classification of unknown metabolites using high-resolution fragmentation mass spectra

K Dührkop, LF Nothias, M Fleischauer, R Reher… - Nature …, 2021 - nature.com
Metabolomics using nontargeted tandem mass spectrometry can detect thousands of
molecules in a biological sample. However, structural molecule annotation is limited to …

Reproducible molecular networking of untargeted mass spectrometry data using GNPS

AT Aron, EC Gentry, KL McPhail, LF Nothias… - Nature protocols, 2020 - nature.com
Abstract Global Natural Product Social Molecular Networking (GNPS) is an interactive online
small molecule–focused tandem mass spectrometry (MS2) data curation and analysis …

Advances in decomposing complex metabolite mixtures using substructure-and network-based computational metabolomics approaches

MA Beniddir, KB Kang, G Genta-Jouve, F Huber… - Natural product …, 2021 - pubs.rsc.org
Covering: up to the end of 2020 Recently introduced computational metabolome mining
tools have started to positively impact the chemical and biological interpretation of …

Indole-containing natural products 2019–2022: isolations, reappraisals, syntheses, and biological activities

SM Umer, M Solangi, KM Khan, RSZ Saleem - Molecules, 2022 - mdpi.com
Indole alkaloids represent a large subset of natural products, with more than 4100 known
compounds. The majority of these alkaloids are biologically active, with some exhibiting …

Natural product anticipation through synthesis

BE Hetzler, D Trauner, AL Lawrence - Nature Reviews Chemistry, 2022 - nature.com
Natural product synthesis remains one of the most vibrant and intellectually rewarding areas
of chemistry, although the justifications for pursuing it have evolved over time. In the early …

Rapid discovery of two unprecedented meroterpenoids from Daphne altaica Pall. using molecular networking integrated with MolNetEnhancer and Network …

WY Zhou, ZH Xi, NN Du, L Ye, MH Jiang, JL Hao… - Chinese Chemical …, 2024 - Elsevier
Under the guidance of the approach which integrates molecular networking,
MolNetEnhancer and Network Annotation Propagation (NAP), daphnaltaicanoids A and B (1 …

Integrated annotation prioritizes metabolites with bioactivity in inflammatory bowel disease

A Bhosle, S Bae, Y Zhang, E Chun… - Molecular Systems …, 2024 - embopress.org
Microbial biochemistry is central to the pathophysiology of inflammatory bowel diseases
(IBD). Improved knowledge of microbial metabolites and their immunomodulatory roles is …

Chemical proportionality within molecular networks

D Petras, AM Caraballo-Rodríguez… - Analytical …, 2021 - ACS Publications
Molecular networking of non-targeted tandem mass spectrometry data connects structurally
related molecules based on similar fragmentation spectra. Here, we report the Chem ical …