Contribution to the Synthesis, Characterization, Separation and Quantification of New N-Acyl Thiourea Derivatives with Antimicrobial and Antioxidant Potential

R Roman, L Pintilie, DC Nuță, MT Căproiu… - Pharmaceutics, 2023 - mdpi.com
The present study aimed to synthesize, characterize, and validate a separation and
quantification method of new N-acyl thiourea derivatives (1a–1o), incorporating thiazole or …

Functionally substituted 2-aminothiazoles as antimicrobial agents: in vitro and in silico evaluation

A Petrou, V Kartsev, A Geronikaki… - SAR and QSAR in …, 2023 - Taylor & Francis
Nine new functionally substituted derivatives of 2-aminothiazole were evaluated for
antimicrobial activity using microdilution method against the panel of eight bacterial and …

Relativistic two-component density functional study of ethyl 2-(2-Iodobenzylidenehydrazinyl) thiazole-4-carboxylate

MW Baig, H Mehmood, T Akhtar - Computational and Theoretical …, 2024 - Elsevier
Relativistic two-component density functional theory employing sf-X2C-S-TD-DFT/SOC
method has been used to explore the detailed electronic spectra of molecules with thiazole …

Synthesis, antimicrobial activity, and biofilm inhibition studies of 1, 2, 3-triazole-containing 2, 3-dihydrothiazole

AA Sediek, AF Kassem, MS Abdel-Aziz… - Synthetic …, 2024 - Taylor & Francis
Abstract The newly synthesized 1, 2, 3-triazole-thiazole hybrids were first evaluated for their
antimicrobial activity against different microbial strains. Most of it showed a marked …

Design, Synthesis of 3‐(Aryl)‐1‐(2‐p‐tolylthiazol‐4‐yl)prop‐2‐en‐1‐ones as Alpha(α)‐Amylase Inhibitors

H Iqbal, M Haroon, T Akhtar, A Aktaş - Chemistry & Biodiversity, 2024 - Wiley Online Library
Abstract α‐Amylase inhibition is vital in controlling diabetic complications. Herein, we have
synthesized a hybrid scaffold based on thiazole‐chalcone to access α‐amylase inhbition …

Design, Synthesis, Anti-Microbial Evaluation, and Docking Studies of New N-Benzyl-3-Indole Derivatives

AA Sediek, AA Shaddy, MAA Radwan… - Egyptian Journal of …, 2024 - ejchem.journals.ekb.eg
New 3-hydrazinecarbothioamide-N-benzylindol derivatives 3a/b have been synthesized by
the reaction of N-benzyl-3-acetylindol 1 with hydrazinecarbothioamide 2a/b. Then …

Synthesis and Characterization of Novel Phthalazin-1 (2H)-one Hybrids with Anticipated Antibacterial Activity

AK Mourad, AY Soliman, AA Makhlouf… - Egyptian Journal of …, 2024 - journals.ekb.eg
Herein, a phthalazine acetohydrazide derivative 4 was assembled and its behaviour
towards carbon nucleophiles was thoroughly investigated. Subsequently, phthalazine …

[PDF][PDF] AJ Csian OURNALOF HEMISTRY AJ Csian OURNALOF HEMISTRY

B POSINASETTY, RK KUMARACHARI… - Asian Journal of …, 2024 - researchgate.net
This study emphasizes the synthesis and characterization of a novel series of oxa cyano
pyridine heterocyclic molecular hybrids (OCP 1-6), integrating pyridine and benzofuran …

Sinteza novih 1, 3-tiazolo-stilbena kao potencijalnih inhibitora kolinesteraza i antioksidansa

L Živko - 2023 - repozitorij.unizg.hr
Sažetak U cilju daljnjeg napredovanja na području sinteze spojeva koji će imati inhibicijsko
djelovanje prema enzimima kolinesterazama i antioksidacijsko djelovanje, sintetizirani su …