A procedure on palladium‐catalyzed carbonylative reaction of trifluoroacetimidoyl chlorides
and nitro compounds for the construction of pharmaceutically valuable 2‐(trifluoromethyl) …

This highlight is the second installment of a series of highlights on nonprecious-metal-
catalyzed reactions of interest to the pharmaceutical industry. Selected transformations from …

A protocol for a copper-catalyzed intermolecular cross-coupling cascade between 2-(2-
bromoaryl)-1 H-benzo [d] imidazole analogues and proline or pipecolic acid has been …

A metal-free and efficient procedure for the synthesis of pyrrolo [1, 2-a] quinoxalines,
quinazolinones, and indolo [1, 2-a] quinoxaline has been developed. The key features of our …

The total synthesis of cyclotripeptidic natural products possessing a central piperazino [2, 1-
b] quinazolin-3, 6-dione core is described through an original strategy involving the pivotal …

The merging of visible-light photoredox and acid catalysis allowed for an intramolecular
Povarov cycloaddition reaction using eosin Y as the photocatalyst and TsOH· H2O as the co …

A three-component reaction catalyzed by base was established, which mainly consisted of
ynals, isocyanates, amines and alcohols. This strategy provides a wide range of substrates …

An efficient and facile approach for the synthesis of quinazolin-4 (3 H)-ones via the reaction
of quinazoline-3-oxides with primary amines is described. This approach is demonstrated to …

Herein, we report the first protocol for visible-light-induced radical isocyanide insertion
reactions between 3-(2-isocyanobenzyl)-indoles and bromodifluoroacetates or …

In this work, an efficient synthesis of indole derivatives through palladium‐catalyzed double
isocyanide insertion reactions has been developed. The reaction intermediates could be …