This review provides a broad perspective of the uses of amino acid fluorides in the synthesis
of peptides and a wide range of other molecules. The topic is discussed with reference to the …

Acid chlorides as peptide coupling agents have its origin in Emil Fischer's era with the first
report of N-protected dipeptide of glycine synthesis emerging in 1903 by Emil Fischer. 1 …

The synthesis of hydroxamic acids starting from carboxylic acids employing 1-
propanephosphonic acid cyclic anhydride (T3P) activation is described. Application of …

The Ugi‐azide reaction of an enantiopure amino acid derived isocyanides, amino acid
esters, aldehydes and TMS‐N3 in MeOH: THF solvent system at 50° C yielded …

The deprotonation of hydrochloride salts of ethyl and methyl esters of amino acids and
peptides is accomplished using activated zinc dust. The reaction is neat and quantitative …

The new cobalt (III) and nickel (II) complexes of the type [M (L) 2 (H 2 O) 2] n+(where M= Co
(III) or Ni (II) ion, n= 3 for Co and 2 for Ni, L= peptides Fmoc. Ala-val-OH (F-AVOH), Fmoc …

Indium-mediated coupling reactions of acyl chlorides and amines for the synthesis of amide
bonds are described. The reaction afforded high yields of the desired amides under mild …

The synthesis of Fmoc amino acid azides starting from the corresponding protected amino
acid and sodium azide (NaN3) by the mixed anhydride method using isobutoxycarbonyl …

Incorporation of the extremely hindered amino acid N-benzylaminoisobutyric acid into
dipeptides under microwave irradiation with commercial zinc dust is described. A …

An efficient and straightforward approach for the coupling of N α-protected hydroxamic acids
with an amino component in the presence of iodine is delineated. The reaction is mediated …