Vicinal diamino functionalities as privileged structural elements in biologically active compounds and exploitation of their synthetic chemistry
SRS Saibabu Kotti, C Timmons… - Chemical biology & drug …, 2006 - Wiley Online Library
The chemistry, synthetic routes and medicinal properties of vicinal diamines and
imidazolines are discussed. Synthetic routes towards chemically and pharmaceutically …
imidazolines are discussed. Synthetic routes towards chemically and pharmaceutically …
Aziridines in formal [3+ 2] cycloadditions: Synthesis of five‐membered heterocycles
AL Cardoso, TMVD Pinho e Melo - European Journal of …, 2012 - Wiley Online Library
Chemistry based on ring opening of aziridines has been widely studied in organic synthesis.
However, it has mainly been centered on ring opening by nucleophiles and on cycloaddition …
However, it has mainly been centered on ring opening by nucleophiles and on cycloaddition …
Nickel-Catalyzed Cross-Electrophile Ring Opening/gem-Difluoroallylation of Aziridines
W Tang, P Fan - Organic Letters, 2023 - ACS Publications
Herein we report a nickel-catalyzed regioselective cross-electrophile ring opening reaction
of sulfonyl-protected aziridines with trifluoromethyl-substituted alkenes as the gem …
of sulfonyl-protected aziridines with trifluoromethyl-substituted alkenes as the gem …
Magic Blue-Initiated SN2-Type Ring Opening of Activated Aziridines: Friedel–Crafts-Type Alkylation of Electron-Rich Arenes/Heteroarenes
A transition metal-free, atom-economical, and highly stereospecific synthetic approach to
Friedel–Crafts-type alkylation of arenes/heteroarenes has been developed. The protocol …
Friedel–Crafts-type alkylation of arenes/heteroarenes has been developed. The protocol …
BF3·OEt2-Mediated Highly Regioselective SN2-Type Ring-Opening of N-Activated Aziridines and N-Activated Azetidines by Tetraalkylammonium Halides
MK Ghorai, A Kumar, DP Tiwari - The Journal of organic chemistry, 2010 - ACS Publications
A highly regioselective Lewis acid-mediated SN2-type ring-opening of N-sulfonylaziridines
and azetidines with tetraalkylammonium halides in CH2Cl2 solution to afford 1, 2-and 1, 3 …
and azetidines with tetraalkylammonium halides in CH2Cl2 solution to afford 1, 2-and 1, 3 …
Stereoselective Lewis Acid Mediated (3+2) Cycloadditions of N‐H‐ and N‐Sulfonylaziridines with Heterocumulenes
RA Craig, NR O'Connor, AFG Goldberg… - … –A European Journal, 2014 - Wiley Online Library
Alkyl and aryl isothiocyanates and carbodiimides are effective substrates in (3+ 2)
cycloadditions with N‐sulfonyl‐2‐substituted aziridines and 2‐phenylaziridine for the …
cycloadditions with N‐sulfonyl‐2‐substituted aziridines and 2‐phenylaziridine for the …
Syntheses of chiral β-and γ-amino ethers, morpholines, and their homologues via nucleophilic ring-opening of chiral activated aziridines and azetidines
MK Ghorai, D Shukla… - The Journal of Organic …, 2012 - ACS Publications
Lewis acid catalyzed quaternary ammonium salt mediated highly regioselective ring-
opening of chiral activated aziridines and azetidines with alcohols to nonracemic β-and γ …
opening of chiral activated aziridines and azetidines with alcohols to nonracemic β-and γ …
Lewis acid catalyzed highly stereoselective domino-ring-opening cyclization of activated aziridines with enolates: synthesis of functionalized chiral γ-lactams
MK Ghorai, DP Tiwari - The Journal of Organic Chemistry, 2010 - ACS Publications
A highly enantio-and diastereoselective Lewis acid catalyzed SN2-type ring opening
followed by cyclization of aziridines with active methylene carbon nucleophiles to …
followed by cyclization of aziridines with active methylene carbon nucleophiles to …
Recent advances in the transformations of cycloalkane-fused oxiranes and aziridines
This account highlights the most relevant transformations of cycloalkane-fused oxiranes and
aziridines developed during the past decade with the intention to provide an overview of the …
aziridines developed during the past decade with the intention to provide an overview of the …
AgSbF6-Promoted Cycloaddition Reaction of 2-Trifluoromethyl-N-tosylaziridine with Aldehydes
R Maeda, R Ishibashi, R Kamaishi, K Hirotaki… - Organic …, 2011 - ACS Publications
AgSbF6-Promoted Cycloaddition Reaction of 2-Trifluoromethyl-N-tosylaziridine with
Aldehydes | Organic Letters ACS ACS Publications C&EN CAS Find my institution Log In …
Aldehydes | Organic Letters ACS ACS Publications C&EN CAS Find my institution Log In …