Role for the propofol hydroxyl in anesthetic protein target molecular recognition

KA Woll, BP Weiser, Q Liang, T Meng… - ACS chemical …, 2015 - ACS Publications
Propofol is a widely used intravenous general anesthetic. We synthesized 2-fluoro-1, 3-
diisopropylbenzene, a compound that we call “fropofol”, to directly assess the significance of …

Discovery of a novel general anesthetic chemotype using high-throughput screening

AR McKinstry-Wu, W Bu, G Rai, WA Lea… - …, 2015 - pubs.asahq.org
Background: The development of novel anesthetics has historically been a process of
combined serendipity and empiricism, with most recent new anesthetics developed via …

[HTML][HTML] Antagonism of Propofol Anesthesia by Alkyl-fluorobenzene Derivatives

DM Plasencia, LH Rodgers, AR Knighton… - Research …, 2024 - ncbi.nlm.nih.gov
Despite their frequent use across many clinical settings, general anesthetics are
medications with lethal side effects and no reversal agents. A fluorinated analogue of …

[PDF][PDF] Antagonism of Propofol Anesthesia by Alkyl-uorobenzene Derivatives

DM Plasencia, LH Rodgers, AR Knighton… - assets-eu.researchsquare.com
Despite their frequent use across many clinical settings, general anesthetics are
medications with lethal side effects and no reversal agents. A fluorinated analogue of …