Synthesis, theoretical properties using DFT method, and nonlinear optical properties of 4-methyl umbelliferone derivative

A Adil, QMA Hassan, TA Alsalim, HA Sultan… - Optik, 2023 - Elsevier
methyl umbelliferone compound is synthesized from resorcinol with ethyl acetoacetate
under ultrasound irradiation as an assistant of reaction. The coumarin derivative, COM-ester …

Identification of novel NLRP3 inhibitors: A comprehensive approach using 2D-QSAR, molecular docking, molecular dynamics simulation and drug-likeness evaluation

M Mouhsin, O Abchir, FS El Otmani, AA Oumghar… - Chemical Papers, 2024 - Springer
This research, employing computational methodologies, aimed to discover potential
inhibitors for the nucleotide-binding oligomerization domain-like receptor protein 3 (NLRP3) …

[HTML][HTML] Synthetic mono-carbonyl curcumin analogues attenuate oxidative stress in mouse models

H Hussain, S Ahmad, SWA Shah, A Ullah, SU Rahman… - Biomedicines, 2022 - mdpi.com
Alzheimer's disease is the commonest form of dementia associated with short-term memory
loss and impaired cognition and, worldwide, it is a growing health issue. A number of …

Prediction of polydimethylsiloxane-water partition coefficients based on the pp-LFER and QSAR models

T Zhu, W Chen, H Cheng, Y Wang, RP Singh - … and Environmental Safety, 2019 - Elsevier
Obtaining accurate measurements of the partition coefficients between sorbent materials
and water is of major importance for the analysis of the adsorption behavior and dissolved …

[HTML][HTML] In-silico modelling studies on some C14-urea-tetrandrine derivatives as potent anti-cancer agents against prostate (PC3) cell line

M Abdullahi, A Uzairu, GA Shallangwa… - Journal of King Saud …, 2020 - Elsevier
Insilico modelling studies was executed on twenty-four (24) novel C 14-urea-tetrandrine
compounds as inhibitors of prostate cancer (PC3) cell line. The molecular structure of each …

[HTML][HTML] Molecular design of curcumin analogues with potent antioxidant properties and thermodynamic evaluation of their mechanism of free radical scavenge

IO Alisi, A Uzairu, SE Abechi - Bulletin of the National Research Centre, 2020 - Springer
Background Free radical attack of cellular structures in the human system is the major cause
of various forms of degenerative diseases. Consequently, recent research has been focused …

QSAR studies on some C14-urea tetrandrine compounds as potent anti-cancer against leukemia cell line (K562)

A Mustapha, G Shallangwa, MT Ibrahim… - Journal of the Turkish …, 2018 - dergipark.org.tr
This research applied Quantitative Structure Activity Relationship (QSAR) technique in
developing a Multiple-Linear Regression (MLR) model using Genetic Functional Algorithm …

[PDF][PDF] A study on hydrogen peroxide scavenging activity and ferric reducing ability of simple coumarins

N Prahadeesh, M Sithambaresan, U Mathiventhan - Emerg. Sci. J, 2018 - academia.edu
Coumarin compounds are δ-lactones where α-pyrone ring is fused with benzene ring.
Coumarins are widely distributed in the plant kingdom as well as they are very important in …

QSAR modelling and docking analysis of some thiazole analogues as alfa-glucosidase inhibitors

MT Ibrahim, A Uzairu, GA Shallangwa… - The Journal of …, 2019 - periodicos.ufv.br
QSAR modelling and docking studies on 45 thiazole analogues were carried out. The
studied compounds in this research were optimized adopting DFT method at B3LYP function …

QSPR modelling for intrinsic viscosity in polymer–solvent combinations based on density functional theory

S Wang, M Cheng, L Zhou, Y Dai… - SAR and QSAR in …, 2021 - Taylor & Francis
Linear and nonlinear quantitative structure–property relationship (QSPR) models were
developed based on a dataset with 65 polymer-solvent combinations. Seven quantum …