Computer-aided prediction of biological activity spectra for organic compounds: The possibilities and limitations

VV Poroikov, DA Filimonov, TA Gloriozova… - Russian Chemical …, 2019 - Springer
We describe the current version of the PASS program for prediction of biological activity
spectra of organic compounds based on analysis of structure—activity relationships (SAR) …

Anthra[1,2-d][1,2,3]triazine-4,7,12(3H)-triones as a New Class of Antistaphylococcal Agents: Synthesis and Biological Evaluation

V Zvarych, M Stasevych, V Novikov, E Rusanov… - Molecules, 2019 - mdpi.com
The development and spread of resistance of human pathogenic bacteria to the action of
commonly used antibacterial drugs is one of the key problems in modern medicine. One of …

9, 10-Anthraquinone dithiocarbamates as potential pharmaceutical substances with pleiotropic actions: Computerized prediction of biological activity and …

MV Stasevich, VI Zvarich, VP Novikov… - Pharmaceutical …, 2020 - Springer
The pleiotropic pharmacological actions of 9, 10-anthraquinone dithiocarbamates were
studied. The Way2Drug web portal was used to establish that cytotoxic, antiviral, and …

Use of impedance biotesting to assess the actions of pharmaceutical compounds on the growth of microorganisms

VS Sibirtsev, IA Naumov, EE Kuprina… - Pharmaceutical …, 2016 - Springer
A method for the analysis of microbial “growth curves” by real-time recording of changes in
the impedance electrical conductance of the medium from multiple samples in parallel is …

[PDF][PDF] Synthesis and antimicrobial activity of nitrogen-containing anthraquinone derivatives

V Shupeniuk, T Taras, O Sabadakh… - Iraqi Journal of …, 2022 - iasj.net
New substituted anthraquinones with amino derivations fragments were synthesized
through the substitution of bromine atom by different amines using the Ullmann coupling …

Efficient amidation of weak amines: synthesis, chiral separation by SFC, and antimicrobial activity of N-(9, 10-dioxo-9, 10-dihydroanthracen-1-yl) carboxamide

K Asokan, AZ Hussain, A Ilangovan - Organic & Biomolecular …, 2024 - pubs.rsc.org
An effective and straightforward method for the synthesis of 1-aminoanthracene-9, 10-dione
carboxamides by coupling a weakly reactive amine, 1-aminoanthracene-9, 10-dione, and …

[PDF][PDF] Synthesis and study of antimicrobial activity of 2-dithiocarbamate-N-(9, 10-dioxo-9, 10-dihydroanthracenyl) acetamides

V Zvarych, M Stasevych… - … Research in Applied …, 2021 - biointerfaceresearch.com
The global emergence and dissemination of multidrug-resistant fungal and bacterial
pathogens is a serious public health threat. The development of novel highly active …

[PDF][PDF] A Computational Approach in the Search of New Biologically Active 9, 10-Anthraquinone Derivatives.

M Stasevych, V Zvarych, V Novikov - IDDM, 2020 - easychair.org
EasyChair Preprint A Computational Approach in the Search of New Biologically Active 9,10-Anthraquinone
Derivatives Page 1 EasyChair Preprint № 4264 A Computational Approach in the Search of …

Кондуктометрическое биотестирование в применении к оценке про-и антибактериальных свойств католитов и анолитов

ВС Сибирцев, АЮ Кулаков… - … технологий, механики и …, 2016 - cyberleninka.ru
Представлена методика применения кондуктометрического биотестирования к
анализу прои антибактериальной активности растворов католита и анолита. При этом …

[PDF][PDF] The new 1, 2, 3-triazolylantracene-9, 10-diones: synthesis and computer bioactivity screening

M Stasevych, V Zvarych, V Lunin, M Vovk… - Chemistry and …, 2017 - researchgate.net
The reactions of 1, 4 (1, 5)-diazido-9, 10-anthracenediones with phenylacetylene and methyl
propiolate under copper (I)-catalyzed reaction of the azidealkyne cycloaddition conditions …