Design, Synthesis, Molecular Docking, Molecular Dynamics and In Vivo Antimalarial Activity of New Dipeptide‐Sulfonamides
A new series of novel dipeptide sulfonamide analogues were designed, synthesized, and
screened for their in silico studies and in vivo antimalarial activities. The synthesized …
screened for their in silico studies and in vivo antimalarial activities. The synthesized …
Design, Synthesis, Molecular Docking, Drug-Likeness/ADMET and Molecular Dynamics Studies of Thiazolyl Benzenesulfonamide Carboxylates as Antimalarial …
In this work, nine novel thiazole derivatives of substituted benzenesulfonamide carboxylate
were designed, synthesized and characterized (1H NMR, 13C NMR and Mass Spectra) for …
were designed, synthesized and characterized (1H NMR, 13C NMR and Mass Spectra) for …
Synthesis, in silico studies and investigations on antimicrobial, antimalarial activities of p-toluenesulphonamoyl 'Leu-Gly'dipeptide carboxamide derivatives
Six novel leucine-glycine dipeptide sulphonamide deriavtives were synthesized and
characterized via 1 HNMR, 13 CNMR, FTIR and HRMS spectroscopic techniques. The in …
characterized via 1 HNMR, 13 CNMR, FTIR and HRMS spectroscopic techniques. The in …
A novel bioinformatic method for the identification of antimicrobial peptides in metagenomes
J Megaw, T Skvortsov, G Gori, AI Dabai… - Journal of Applied …, 2024 - academic.oup.com
Aims This study aimed to develop a new bioinformatic approach for the identification of
novel antimicrobial peptides (AMPs), which did not depend on sequence similarity to known …
novel antimicrobial peptides (AMPs), which did not depend on sequence similarity to known …
Effect of Leu/Val mutation on the energetics of antimicrobial peptide: micelle binding
S Ghosh, S Chatterjee, P Satpati - The Journal of Physical …, 2022 - ACS Publications
Recently, we had reported a synthetic positively charged leucine-rich 14-residue-long
antimicrobial peptide (AMP, LL-14: NH3+-LKWLKKLLKWLKKL-CONH2), which was highly …
antimicrobial peptide (AMP, LL-14: NH3+-LKWLKKLLKWLKKL-CONH2), which was highly …
New substituted benzenesulphonamoyl 'Cys-Gly'dipeptide carboxamide derivatives: Design, synthesis, characterization and pharmacological studies
Abstract Twelve new sulphonamide (Cys-Gly) dipeptide carboxamide derivatives 17a–17l
were designed, prepared and characterized through spectroscopic techniques and their …
were designed, prepared and characterized through spectroscopic techniques and their …
Evaluation of glycyl-arginine and lysyl-aspartic acid dipeptides for their antimicrobial, antibiofilm, and anticancer potentials
Antibacterial resistance and cancer are worldwide challenges and have been defined as
major threats by international health organizations. Peptides are produced naturally by all …
major threats by international health organizations. Peptides are produced naturally by all …
Synthesis and Biological Evaluation of Dipeptide-Based Stilbene Derivatives Bearing a Biheterocyclic Moiety as Potential Fungicides
Y Zhu, X Lin, L Wen, D He - Molecules, 2022 - mdpi.com
The escalating demand for crop production, environmental protection, and food safety
warrants the development of new fungicides with greater efficiency, environmental …
warrants the development of new fungicides with greater efficiency, environmental …
Antimicrobial, Antibiofilm and Anticancer Potentials of Glycine and Glycyl-Glycine; an in vitro study
Globally, there is a huge demand for novel agents capable of providing protection against
both pathogen microorganisms and tumor cells. In this study, the antimicrobial, biofilm …
both pathogen microorganisms and tumor cells. In this study, the antimicrobial, biofilm …
[PDF][PDF] Antimicrobial, Antibiofilm and Anticancer Potentials of Glycine and Glycyl-Glycine; an in vitro study Glisin ve Glisil-Glisinin Antimikrobiyal, Antibiyofilm ve …
ÖZ Küresel anlamda, hem patojen mikroorganizmalara karşı koruma sağlayabilen hem de
tümör hücrelerine karşı etkili olabilen yeni ajanlara karşı büyük bir talep bulunmaktadır. Bu …
tümör hücrelerine karşı etkili olabilen yeni ajanlara karşı büyük bir talep bulunmaktadır. Bu …