One-pot, three-component assembly of indoloquinolines: Total synthesis of isocryptolepine
AV Aksenov, DA Aksenov, NA Orazova… - The Journal of …, 2017 - ACS Publications
Indolo [3, 2-c] quinolones have been efficiently synthesized via an acid-mediated, one-pot,
three-component condensation of arylhydrazines, o-aminoacetophenones, and triazines or …
three-component condensation of arylhydrazines, o-aminoacetophenones, and triazines or …
Substituted isoquinolinones and quinazolinones
J Berghausen, N Buschmann, P Furet… - US Patent …, 2013 - Google Patents
2011-04-26 Assigned to NOVARTIS AG reassignment NOVARTIS AG ASSIGNMENT OF
ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors: HERGOVICH …
ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors: HERGOVICH …
Synthesis and contractile activity of substituted 1, 2, 3, 4-tetrahydroisoquinolines
A series of different 1-monosubstituted and 1, 1-disubstituted 1, 2, 3, 4-tetrahydro-
isoquinolines was synthesized in high yields from different ketoamides. We have developed …
isoquinolines was synthesized in high yields from different ketoamides. We have developed …
Substituted isoquinolinones and quinazolinones
J Berghausen, N Buschmann, P Furet… - US Patent …, 2015 - Google Patents
0 [3*] N ([3*]) C (= O) C (C) C.[3*] N ([3*]) C (= O) C (C) C (C) C.[3*] N ([3*]) C (C) C (C) C.[3*]
N ([3*]) C1 (C (C) C) CC1.[3*] N ([3*]) CC (C) C (C) C Chemical compound [3*] N ([3*]) C …
N ([3*]) C1 (C (C) C) CC1.[3*] N ([3*]) CC (C) C (C) C Chemical compound [3*] N ([3*]) C …
Crystalline form of an inhibitor of MDM2/4 and p53 interaction
J Berghausen, REN Haixia - US Patent 9,073,898, 2015 - Google Patents
(57) ABSTRACT A crystalline form of (S)-1-(4-Chloro-phenyl)-7-isopropoxy 6-methoxy-2-(4-
methyl-4-(4-methyl-3-oxo-piperazin-1-yl)-trans-cyclohexylmethyl-amino-phenyl)-1, 4-dihydro …
methyl-4-(4-methyl-3-oxo-piperazin-1-yl)-trans-cyclohexylmethyl-amino-phenyl)-1, 4-dihydro …
Synthesis of N-[1-(2-Acetyl-4,5-dimethoxyphenyl)propan-2-yl]benzamide and Its Copper(II) Complex
P Marinova, S Nikolova, S Tsoneva - Russian Journal of General …, 2023 - Springer
This paper represents a convenient method for the synthesis of N-[1-(2-acetyl-4, 5-
dimethoxyphenyl) propan-2-yl] benzamide and its Cu (II) complex. In silico analysis …
dimethoxyphenyl) propan-2-yl] benzamide and its Cu (II) complex. In silico analysis …
[PDF][PDF] Molecular iodine oxidative cyclocondesation of ortho-aminobenzamide with aryl aldehydes: A new and efficient access to quinazolin-4 (3H)-ones
M Bakavoli, M Rahimizadeh, A Shiri, Z Ebrahimpour - Iran. J. Org. Chem, 2009 - Citeseer
Molecular iodine oxidative cyclocondesation of ortho-aminobenzamide with aryl aldehydes: A
new and efficient access to quinazoli Page 1 Iranian Journal of Organic Chemistry 1 (2009) …
new and efficient access to quinazoli Page 1 Iranian Journal of Organic Chemistry 1 (2009) …
Crystalline form of an inhibitor of MDM2/4 and p53 interaction
J Berghausen, REN Haixia - US Patent 8,969,351, 2015 - Google Patents
The present invention relates to a crystalline form of (S)-1-(4-Chloro-phenyl)-7-isopropoxy-6-
methoxy-2-(4-me thyl-4-(4-methyl-3-oxo-piperazin-1-yl)-trans-cyclohexyl methyl-amino …
methoxy-2-(4-me thyl-4-(4-methyl-3-oxo-piperazin-1-yl)-trans-cyclohexyl methyl-amino …
[PDF][PDF] Regioselective acylation of β-enaminones of homoveratrylamine
Regioselective acylation of β-enaminones of homoveratrylamine Page 1 General Papers
ARKIVOC 2007 (xv) 11-17 ISSN 1424-6376 Page 11 ©ARKAT USA, Inc. Regioselective …
ARKIVOC 2007 (xv) 11-17 ISSN 1424-6376 Page 11 ©ARKAT USA, Inc. Regioselective …
Pyrrolopyrrolone derivatives and their use as BET inhibitors
H Rueger, J Blank, V Bordas, S Cotesta, G Bold… - US Patent …, 2017 - Google Patents
2016-07-16 Assigned to NOVARTIS PHARMA AG reassignment NOVARTIS PHARMA AG
ASSIGNMENT OF ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors …
ASSIGNMENT OF ASSIGNORS INTEREST (SEE DOCUMENT FOR DETAILS). Assignors …