Neurosteroid receptor modulators for treating traumatic brain injury

TA Verdoorn, TJ Parry, G Pinna, J Lifshitz - Neurotherapeutics, 2023 - Elsevier
Traumatic brain injury (TBI) triggers wide-ranging pathology that impacts multiple
biochemical and physiological systems, both inside and outside the brain. Functional …

Exploring the Transmembrane Allostery in MexB: DB08385 Variant as Promising Inhibitor like Candidate Against Pseudomonas aeruginosa Antibiotic Resistance–A …

A Bera, S Mukherjee, N Patra - Physical Chemistry Chemical Physics, 2024 - pubs.rsc.org
Pseudomonas aeruginosa, a formidable pathogen renowned for its antimicrobial resistance,
poses a significant threat to immunocompromised individuals. In that respect, the MexAB …

Improving the Solubility and Bioavailability of Progesterone Cocrystals with Selected Carboxylic Acids

J Xiong, D Xu, H Zhang, Y Shi, X Wu, S Wang - Pharmaceutics, 2024 - mdpi.com
Progesterone (PROG) is a natural steroid hormone with low solubility and high permeability
that belongs to biopharmaceutics classification system class II. In this study, novel …

Amine‐Carbamate Self‐Immolative Spacers Counterintuitively Release 3° Alcohol at Much Faster Rates than 1° Alcohol Payloads

M Mason, L Bisbal Lopez, F Bashiri, A Herrero… - …, 2024 - Wiley Online Library
Self‐immolative (SI) spacers are degradable chemical connectors widely used in prodrugs
and drug conjugates to release pharmaceutical ingredients in response to specific stimuli …

Microglial polarization pathways and therapeutic drugs targeting activated microglia in traumatic brain injury

L Shi, S Liu, J Chen, H Wang, Z Wang - Neural Regeneration Research - journals.lww.com
Traumatic brain injury can be categorized into primary and secondary injuries. Secondary
injuries are the main cause of disability following traumatic brain injury, which involves a …