Recent progress in cyclic aryliodonium chemistry: syntheses and applications
X Peng, A Rahim, W Peng, F Jiang, Z Gu… - Chemical …, 2023 - ACS Publications
Hypervalent aryliodoumiums are intensively investigated as arylating agents. They are
excellent surrogates to aryl halides, and moreover they exhibit better reactivity, which allows …
excellent surrogates to aryl halides, and moreover they exhibit better reactivity, which allows …
A minireview of 1, 2, 3‐triazole hybrids with O‐heterocycles as leads in medicinal chemistry
Over the past few decades, the dynamic progress in the synthesis and screening of
heterocyclic compounds against various targets has made a significant contribution in the …
heterocyclic compounds against various targets has made a significant contribution in the …
New 1, 3, 4‐oxadiazoles linked with the 1, 2, 3‐triazole moiety as antiproliferative agents targeting the EGFR tyrosine kinase
Abstract A series of 1, 3, 4‐oxadiazole‐1, 2, 3‐triazole hybrids bearing different
pharmacophoric moieties has been designed and synthesized. Their antiproliferative activity …
pharmacophoric moieties has been designed and synthesized. Their antiproliferative activity …
Synthesis of vanillin derivatives with 1, 2, 3‐triazole fragments and evaluation of their fungicide and fungistatic activities
PAR Gazolla, AR de Aguiar, MCA Costa… - Archiv der …, 2023 - Wiley Online Library
Vanillin is the main component of natural vanilla extract and is responsible for its flavoring
properties. Besides its well‐known applications as an additive in food and cosmetics, it has …
properties. Besides its well‐known applications as an additive in food and cosmetics, it has …
MOF-Derived Cu@ NC Catalyst for 1, 3-Dipolar Cycloaddition Reaction
Z Wang, X Zhou, S Gong, J Xie - Nanomaterials, 2022 - mdpi.com
Cu (im) 2-derived Cu@ NC composites were used for the first time as efficient
heterogeneous catalysts for one-pot 1, 3-dipolar cycloaddition of terminal alkynes, aryl …
heterogeneous catalysts for one-pot 1, 3-dipolar cycloaddition of terminal alkynes, aryl …
Synthesis and anticancer activity of 3-(1-aryl-5-methyl-1H-1, 2, 3-triazol-4-yl)-1-phenyl-1H-pyrazole-4-carbaldehydes
BF Abdel-Wahab, BM Kariuki, HA Mohamed… - Journal of Molecular …, 2023 - Elsevier
The generation of heterocycles containing 1, 2, 3-triazole and pyrazole moieties has been
explored. The synthesis of these heterocycles is of interest because they are components of …
explored. The synthesis of these heterocycles is of interest because they are components of …
Ligand-Based Pharmacophoric Design and Anti-inflammatory Evaluation of Triazole Linked Semisynthetic Labdane Conjugates
S Mohan, L Krishnan, N Madhusoodanan… - ACS Medicinal …, 2024 - ACS Publications
This study employed a ligand-based pharmacophoric approach to design and synthesize 33
novel semisynthetic labdane-appended triazolyl isatins to discover potential anti …
novel semisynthetic labdane-appended triazolyl isatins to discover potential anti …
Process-Divergent Syntheses of 4-and 5-Sulfur-Functionalized 1, 2, 3-Triazoles via Copper-Catalyzed Azide–Alkyne Cycloadditions of 1-Phosphinyl-2 …
L Peng, Y Zhao, Y Okuda, L Le, Z Tang… - The Journal of …, 2023 - ACS Publications
4-Sulfanyl-substituted 1, 2, 3-triazoles were provided regioselectively with good yields and
broad scope via consecutive t-BuOK-promoted dephosphinylation of 1-phosphinyl-2 …
broad scope via consecutive t-BuOK-promoted dephosphinylation of 1-phosphinyl-2 …
In Situ-Generated Formamidine as a Carbon/Nitrogen Source for Enaminone Formation: One-Pot Synthesis of Functionalized 4-Acyl-1, 2, 3-triazoles
JX Lin, YX Chen, MC Chien, HJ Chen… - The Journal of …, 2024 - ACS Publications
N, N-Dimethylformamide was reacted with hexamethyldisilazane to generate an N, N-
dimethylformimidamide intermediate; thereafter, a reaction with acetophenones/β-diketones …
dimethylformimidamide intermediate; thereafter, a reaction with acetophenones/β-diketones …
Design, Synthesis, in vitro and in silico Characterization of 2‐Quinolone‐L‐alaninate‐1,2,3‐triazoles as Antimicrobial Agents
Due to the ever‐increasing antimicrobial resistance there is an urgent need to continuously
design and develop novel antimicrobial agents. Inspired by the broad antibacterial activities …
design and develop novel antimicrobial agents. Inspired by the broad antibacterial activities …