Molecular targeted therapy of glioblastoma

E Le Rhun, M Preusser, P Roth, DA Reardon… - Cancer treatment …, 2019 - Elsevier
Glioblastomas are intrinsic brain tumors thought to originate from neuroglial stem or
progenitor cells. More than 90% of glioblastomas are isocitrate dehydrogenase (IDH) …

Function of the c-Met receptor tyrosine kinase in carcinogenesis and associated therapeutic opportunities

Y Zhang, M Xia, K Jin, S Wang, H Wei, C Fan, Y Wu… - Molecular cancer, 2018 - Springer
Abstract c-Met is a receptor tyrosine kinase belonging to the MET (MNNG HOS transforming
gene) family, and is expressed on the surfaces of various cells. Hepatocyte growth factor …

The landscape of genomic alterations across childhood cancers

SN Gröbner, BC Worst, J Weischenfeldt, I Buchhalter… - Nature, 2018 - nature.com
Pan-cancer analyses that examine commonalities and differences among various cancer
types have emerged as a powerful way to obtain novel insights into cancer biology. Here we …

Integrated molecular meta-analysis of 1,000 pediatric high-grade and diffuse intrinsic pontine glioma

A Mackay, A Burford, D Carvalho, E Izquierdo… - Cancer cell, 2017 - cell.com
We collated data from 157 unpublished cases of pediatric high-grade glioma and diffuse
intrinsic pontine glioma and 20 publicly available datasets in an integrated analysis of> …

MET-dependent solid tumours—molecular diagnosis and targeted therapy

R Guo, J Luo, J Chang, N Rekhtman, M Arcila… - Nature reviews Clinical …, 2020 - nature.com
Attempts to develop MET-targeted therapies have historically focused on MET-expressing
cancers, with limited success. Thus, MET expression in the absence of a genomic marker of …

HGF/c-MET pathway in cancer: from molecular characterization to clinical evidence

J Fu, X Su, Z Li, L Deng, X Liu, X Feng, J Peng - Oncogene, 2021 - nature.com
This review provides a comprehensive landscape of HGF/c-MET (hepatocyte growth factor
(HGF)/mesenchymal–epithelial transition factor (c-MET)) signaling pathway in cancers. First …

Infant high-grade gliomas comprise multiple subgroups characterized by novel targetable gene fusions and favorable outcomes

M Clarke, A Mackay, B Ismer, JC Pickles… - Cancer discovery, 2020 - AACR
Infant high-grade gliomas appear clinically distinct from their counterparts in older children,
indicating that histopathologic grading may not accurately reflect the biology of these tumors …

Mutational landscape of secondary glioblastoma guides MET-targeted trial in brain tumor

H Hu, Q Mu, Z Bao, Y Chen, Y Liu, J Chen, K Wang… - Cell, 2018 - cell.com
Low-grade gliomas almost invariably progress into secondary glioblastoma (sGBM) with
limited therapeutic option and poorly understood mechanism. By studying the mutational …

Known and novel roles of the MET oncogene in cancer: a coherent approach to targeted therapy

PM Comoglio, L Trusolino, C Boccaccio - Nature Reviews Cancer, 2018 - nature.com
The MET oncogene encodes an unconventional receptor tyrosine kinase with pleiotropic
functions: it initiates and sustains neoplastic transformation when genetically altered …

Receptor tyrosine kinases and cancer: oncogenic mechanisms and therapeutic approaches

P Saraon, S Pathmanathan, J Snider, A Lyakisheva… - Oncogene, 2021 - nature.com
Receptor tyrosine kinases (RTKs) are transmembrane receptors of great clinical interest due
to their role in disease, notably cancer. Since their discovery, several mechanisms of RTK …