[HTML][HTML] Emerging trends and future opportunities for coumarin-heterocycle conjugates as antibacterial agents
YF Mustafa - Results in Chemistry, 2023 - Elsevier
Infectious diseases resulting from various strains of pathogenic bacteria are among the
leading causes of death and morbidity worldwide. The currently-available antibacterial …
leading causes of death and morbidity worldwide. The currently-available antibacterial …
Relationship between Structure and Antibacterial Activity of α-Aminophosphonate Derivatives Obtained via Lipase-Catalyzed Kabachnik− Fields Reaction
D Koszelewski, P Kowalczyk, P Śmigielski… - Materials, 2022 - mdpi.com
We reported a new method dealing with the synthesis of novel pharmacologically relevant α-
aminophosphonate derivatives via a lipase-catalyzed Kabachnik− Fields reaction with yields …
aminophosphonate derivatives via a lipase-catalyzed Kabachnik− Fields reaction with yields …
Promiscuous Lipase-Catalyzed Knoevenagel–Phospha–Michael Reaction for the Synthesis of Antimicrobial β-Phosphono Malonates
J Samsonowicz-Górski, D Koszelewski… - International Journal of …, 2022 - mdpi.com
An enzymatic route for phosphorous–carbon bond formation was developed by discovering
new promiscuous activity of lipase. We reported a new metal-free biocatalytic method for the …
new promiscuous activity of lipase. We reported a new metal-free biocatalytic method for the …
Enzymatic Synthesis of a Novel Coumarin Aminophosphonates: Antibacterial Effects and Oxidative Stress Modulation on Selected E. coli Strains
D Koszelewski, P Kowalczyk, A Brodzka… - International Journal of …, 2023 - mdpi.com
The objective of the present study was to evaluate the synergistic effect of two important
pharmacophores, coumarin and α-amino dimethyl phosphonate moieties, on antimicrobial …
pharmacophores, coumarin and α-amino dimethyl phosphonate moieties, on antimicrobial …
Influence of Open Chain and Cyclic Structure of Peptidomimetics on Antibacterial Activity in E. coli Strains
P Sahrawat, P Kowalczyk, D Koszelewski, M Szymczak… - Molecules, 2022 - mdpi.com
An efficient method for the synthesis of functionalized peptidomimetics via multicomponent
Ugi reaction has been developed. The application of trifluoroethanol (TFE) as a reaction …
Ugi reaction has been developed. The application of trifluoroethanol (TFE) as a reaction …
Synthesis and Antimicrobial Activity of the Pathogenic E. coli Strains of p-Quinols: Additive Effects of Copper-Catalyzed Addition of Aryl Boronic Acid to …
D Koszelewski, P Kowalczyk… - International Journal of …, 2023 - mdpi.com
A mild and efficient protocol for the synthesis of p-quinols under aqueous conditions was
developed. The pivotal role of additives in the copper-catalyzed addition of aryl boronic and …
developed. The pivotal role of additives in the copper-catalyzed addition of aryl boronic and …
Direct heteroarylation polymerization of a π-conjugated polymer with degradable 1, 2, 4-oxadiazole linkers
BR Varju, DS Seferos - Polymer Chemistry, 2022 - pubs.rsc.org
The synthesis of π-conjugated polymers containing a degradable 1, 2, 4-oxadiazole linker
by direct heteroaryl polymerization (DHAP) is reported. The 1, 2, 4-oxadiazole linker is …
by direct heteroaryl polymerization (DHAP) is reported. The 1, 2, 4-oxadiazole linker is …
The Synthesis and Evaluation of Diethyl Benzylphosphonates as Potential Antimicrobial Agents
A Brodzka, P Kowalczyk, D Trzepizur, D Koszelewski… - Molecules, 2022 - mdpi.com
The impact of substituent at phenyl ring of diethyl benzylphosphonate derivatives on
cytotoxic activity was studied. The organophosphonates were obtained based on developed …
cytotoxic activity was studied. The organophosphonates were obtained based on developed …
Functionalised Anodised Aluminium Oxide as a Biocidal Agent
M Schabikowski, M Laskowska, P Kowalczyk… - International Journal of …, 2022 - mdpi.com
In this article, we describe the antimicrobial properties of a new composite based on anodic
aluminium oxide (AAO) membranes containing propyl-copper-phosphonate units arranged …
aluminium oxide (AAO) membranes containing propyl-copper-phosphonate units arranged …
Aluminium (III) Oxide—The Silent Killer of Bacteria
M Schabikowski, P Kowalczyk, A Karczmarska… - Molecules, 2023 - mdpi.com
In this article, we describe the antimicrobial properties of pristine anodised aluminium oxide
matrices—the material many consider biologically inert. During a typical anodisation …
matrices—the material many consider biologically inert. During a typical anodisation …