Glucocorticosteroids, processes for their preparation, pharmaceutical compositions containing them and their use in therapy
H Bladh, F Burkamp, B Gabos, P Hansen… - US Patent …, 2012 - Google Patents
First worldwide family litigation filed litigation Critical https://patents. darts-ip. com/? family=
40328402&utm_source= google_patent&utm_medium= platform_link&utm_campaign …
40328402&utm_source= google_patent&utm_medium= platform_link&utm_campaign …
Bi-functional pyrazolopyridine compounds
WR Baker, S Cai, JA Kaplan, M Kim, G Phillips… - US Patent …, 2013 - Google Patents
4,992.474. A 2f1991 Skidmore et al. 5,455.252 A 10, 1995 Wilhelmet al. 5,712.298 A 1/1998
Amschler 5,728,712 A 3, 1998 Montana et al. HO 5,776,983 A 7, 1998 Washburn et al …
Amschler 5,728,712 A 3, 1998 Montana et al. HO 5,776,983 A 7, 1998 Washburn et al …
Bi-functional quinoline analogs
WR Baker, S Cai, JA Kaplan, M Kim… - US Patent …, 2013 - Google Patents
US PATENT DOCUMENTS wherein X is: 3,885,047 A 5, 1975 Seidehamel et al. 4,145,542
A 3/1979 Nakagawa et al. 4,761,421 A 8, 1988 Muir 4,992.474. A 2f1991 Skidmore et al. O …
A 3/1979 Nakagawa et al. 4,761,421 A 8, 1988 Muir 4,992.474. A 2f1991 Skidmore et al. O …
Novel compounds
F Burkamp, P Hansen - US Patent App. 12/749,919, 2010 - Google Patents
0002 The present invention relates to compounds having glucocorticosteroid receptor
agonist activity, processes for their preparation, pharmaceutical compositions containing …
agonist activity, processes for their preparation, pharmaceutical compositions containing …
Novel amide compounds
F Burkamp, B Gabos, S Ivanova… - US Patent App. 12 …, 2010 - Google Patents
0002 The present invention relates to compounds having glucocorticosteroid receptor
agonist activity, processes for their preparation, pharmaceutical compositions containing …
agonist activity, processes for their preparation, pharmaceutical compositions containing …
Combination 408
S Connolly, A Fisher, A Humphries… - US Patent App. 12 …, 2010 - Google Patents
The invention provides a pharmaceutical product, kit or com position comprising a first active
ingredient which is N-Cy clohexyl-N'-[2-(3-fluorophenyl) ethyl-N-(2-[2-(4-hy droxy-2-oxo-2, 3 …
ingredient which is N-Cy clohexyl-N'-[2-(3-fluorophenyl) ethyl-N-(2-[2-(4-hy droxy-2-oxo-2, 3 …
Bi-functional pyrazolopyridine compounds
WR Baker, S Cai, JA Kaplan, M Kim, G Phillips… - US Patent …, 2013 - Google Patents
May 9, 2011.(57) ABSTRACT (60) Provisional application No. 61/333,031, filed on May This
invention provides compounds of the formula: 10, 2010, provisional application No …
invention provides compounds of the formula: 10, 2010, provisional application No …
Steroid Derivatives Acting As Glucocorticosteroid Receptor Agonists
0001. The present invention relates to compounds having glucocorticosteroid receptor
agonist activity, processes for their preparation, pharmaceutical compositions containing …
agonist activity, processes for their preparation, pharmaceutical compositions containing …