Current medicinal chemistry relies heavily on the quality of building blocks, ie reagents used
to introduce chemical diversity into the target molecules. The last decade witnessed an …

Sulfonyl fluoride (SF) containing substances are currently attracting enormous attention
among practitioners of both chemical biology and synthetic organic chemistry. The groups of …

SuFEx reactions, in which an S− F moiety reacts with a silyl‐protected phenol, have been
developed as powerful click reactions. In the current paper we open up the potential of …

An up-to-date short review of the chalcone methodologies is presented, which is the most
interesting and beneficial for choosing the desired protocol to synthesize suitable derivatives …

An electrochemistry-promoted oxidative cleavage of (sp3) C–C (sp3)/H bonds in alkylarenes
was developed. Various aryl alkanes can be smoothly converted into ketones/aldehydes …

In this work, we report the anti‐microbial and computational study of two 2, 3‐dihydro‐1 H‐
inden‐1‐one derived fluorinated chalcone scaffolds. The (E)‐2‐(4‐(trifluoromethyl) …

Chemoselective transformations of functionalized sulfonyl fluorides and chlorides are
surveyed comprehensively. It is shown that sulfonyl fluorides provide an excellent selectivity …

Multigram synthesis of (chlorosulfonyl) benzenesulfonyl fluorides is described. Selective
modification of these building blocks at the sulfonyl chloride function under parallel …

A series of quinoline-chalcones were synthesized from one-pot Friedlander annulation
followed by Claisen–Schmidt condensation in the presence of tetrabutylammonium-ionic …

A series of chalcones with various substituents and their novel pyrazole and pyrazoline
derivatives were synthesized. The pyrazole derivatives were synthesized in two ways: via …