An overview on the anticancer activity of Ru (II)/acylthiourea complexes
GH Ribeiro, AR Costa, AR de Souza… - Coordination Chemistry …, 2023 - Elsevier
This review outlines research on the development of ruthenium complexes containing
acylthiourea ligands with potential antitumor activity, which have been leveraged in recent …
acylthiourea ligands with potential antitumor activity, which have been leveraged in recent …
Medicinal importance, coordination chemistry with selected metals (Cu, Ag, Au) and chemosensing of thiourea derivatives. A review
Thiourea and its derivatives are versatile compounds used in several fields of life ranging
from medicinal to chemosensor applications. In this review article, generally used …
from medicinal to chemosensor applications. In this review article, generally used …
Current developments in chemistry, coordination, structure and biological aspects of 1-(acyl/aroyl)-3-(substituted) thioureas: advances Continue…
A Saeed, MN Mustafa, M Zain-ul-Abideen… - Journal of Sulfur …, 2019 - Taylor & Francis
(acyl/aroyl)-3-(substituted) thioureas are exciting structures in the fields of organic synthesis,
material sciences, and biomedical research. Of particular significance is the fact that acyl …
material sciences, and biomedical research. Of particular significance is the fact that acyl …
Design, synthesis, kinetic mechanism and molecular docking studies of novel 1-pentanoyl-3-arylthioureas as inhibitors of mushroom tyrosinase and free radical …
A series of novel 1-pentanoyl-3-arylthioureas was designed as new mushroom tyrosinase
inhibitors and free radical scavengers. The title compounds were obtained in excellent yield …
inhibitors and free radical scavengers. The title compounds were obtained in excellent yield …
New acetylphenol-based acyl thioureas broaden the scope of drug candidates for urease inhibition: synthesis, in vitro screening and in silico analysis
Helicobacter pylori urease remains a validated drug target for the eradication of pervasive
chronic stomach infection that leads to severe human health diseases such as gastritis and …
chronic stomach infection that leads to severe human health diseases such as gastritis and …
Synthesis, molecular docking studies of coumarinyl-pyrazolinyl substituted thiazoles as non-competitive inhibitors of mushroom tyrosinase
A series of coumarinyl-pyrazolinyl substituted thiazoles derivatives were synthesized and
their inhibitory effects on the DPPH and mushroom tyrosinase were evaluated. The results …
their inhibitory effects on the DPPH and mushroom tyrosinase were evaluated. The results …
Novel C-2 symmetric molecules as α-glucosidase and α-amylase inhibitors: design, synthesis, kinetic evaluation, molecular docking and pharmacokinetics
A series of symmetrical salicylaldehyde-bishydrazine azo molecules, 5a–5h, have been
synthesized, characterized by 1H-NMR and 13C-NMR, and evaluated for their in vitro α …
synthesized, characterized by 1H-NMR and 13C-NMR, and evaluated for their in vitro α …
Sulfonamide-linked ciprofloxacin, sulfadiazine and amantadine derivatives as a novel class of inhibitors of jack bean urease; synthesis, kinetic mechanism and …
Sulfonamide derivatives serve as an important building blocks in the drug design discovery
and development (4D) process. Ciprofloxacin-, sulfadiazine-and amantadine-based …
and development (4D) process. Ciprofloxacin-, sulfadiazine-and amantadine-based …
Hybrid pharmacophoric approach in the design and synthesis of coumarin linked pyrazolinyl as urease inhibitors, kinetic mechanism and molecular docking
The current research article reports the synthesis of coumarinyl pyrazolinyl thioamide
derivatives and their biological activity as inhibitors of jack bean urease. The coumarinyl …
derivatives and their biological activity as inhibitors of jack bean urease. The coumarinyl …
Green Synthesis of Gold and Iron Nanoparticles for Targeted Delivery: An In Vitro and In Vivo Study
Nanotechnology has vast applications in almost all fields of science and technology. The
use of medicinal plants for the synthesis of metallic nanoparticles has gained much attention …
use of medicinal plants for the synthesis of metallic nanoparticles has gained much attention …