Targeted therapies for triple-negative breast cancer: combating a stubborn disease

M Kalimutho, K Parsons, D Mittal, JA López… - Trends in …, 2015 - cell.com
Triple-negative breast cancers (TNBCs) constitute a heterogeneous subtype of breast
cancers that have a poor clinical outcome. Although no approved targeted therapy is …

A recent update on small‐molecule kinase inhibitors for targeted cancer therapy and their therapeutic insights from mass spectrometry‐based proteomic analysis

PY Lee, Y Yeoh, TY Low - The FEBS Journal, 2023 - Wiley Online Library
Kinases are key regulatory signalling proteins governing numerous essential biological
processes and cellular functions. Dysregulation of many protein kinases is associated with …

Turning liabilities into opportunities: Off-target based drug repurposing in cancer

V Palve, Y Liao, LLR Rix, U Rix - Seminars in cancer biology, 2021 - Elsevier
Targeted drugs and precision medicine have transformed the landscape of cancer therapy
and significantly improved patient outcomes in many cases. However, as therapies are …

Higher levels of TIMP-1 expression are associated with a poor prognosis in triple-negative breast cancer

G Cheng, X Fan, M Hao, J Wang, X Zhou, X Sun - Molecular cancer, 2016 - Springer
Background Tissue inhibitor of metalloproteinases-1 (TIMP-1) is a multifunctional protein
that can directly regulate apoptosis and metastasis. In this study, we investigated the …

Predicting and overcoming chemotherapeutic resistance in breast cancer

KH Chun, JH Park, S Fan - Translational Research in Breast Cancer …, 2017 - Springer
Our understanding of breast cancer and its therapeutic approach has improved greatly due
to the advancement of molecular biology in recent years. Clinically, breast cancers are …

Targeting epithelial–mesenchymal plasticity in cancer: clinical and preclinical advances in therapy and monitoring

S Bhatia, J Monkman, AKL Toh, SH Nagaraj… - Biochemical …, 2017 - portlandpress.com
The concept of epithelial–mesenchymal plasticity (EMP), which describes the dynamic flux
within the spectrum of phenotypic states that invasive carcinoma cells may reside, is being …

Identification of selective cytotoxic and synthetic lethal drug responses in triple negative breast cancer cells

P Gautam, L Karhinen, A Szwajda, SK Jha, B Yadav… - Molecular cancer, 2016 - Springer
Background Triple negative breast cancer (TNBC) is a highly heterogeneous and
aggressive type of cancer that lacks effective targeted therapy. Despite detailed molecular …

Materials, workflows and applications of IMAC for phosphoproteome profiling in the recent decade: A review

R Tang, Q Bai, S Ma, J Ou - TrAC Trends in Analytical Chemistry, 2023 - Elsevier
The last ten years have witnessed the increasingly notable advances in immobilized metal
ion chromatography (IMAC) for phosphoproteomic profiling. Protein phosphorylation is an …

ANP 32E induces tumorigenesis of triple‐negative breast cancer cells by upregulating E2F1

Z Xiong, L Ye, H Zhenyu, F Li, Y Xiong, C Lin… - Molecular …, 2018 - Wiley Online Library
Triple‐negative breast cancer (TNBC) lacks expression of estrogen receptor (ER),
progesterone receptor, and the HER 2 receptor; it is highly proliferative and becomes the …

[HTML][HTML] Emerging therapies for acute myeloid leukemia: translating biology into the clinic

S Kavanagh, T Murphy, A Law, D Yehudai, JM Ho… - JCI insight, 2017 - ncbi.nlm.nih.gov
Acute myeloid leukemia (AML) is an aggressive hematological malignancy with a poor
outcome; overall survival is approximately 35% at two years and some subgroups have a …