Modified curcumins as potential drug candidates for breast cancer: An overview

AL Flint, DW Hansen, LVD Brown, LE Stewart, E Ortiz… - Molecules, 2022 - mdpi.com
Breast cancer (BC), the most common malignancy in women, results from significant
alterations in genetic and epigenetic mechanisms that alter multiple signaling pathways in …

Recent advances of curcumin derivatives in breast cancer

Y Yin, Y Tan, X Wei, X Li, H Chen, Z Yang… - Chemistry & …, 2022 - Wiley Online Library
Curcumin is a potential plant‐derived drug for the treatment of breast cancer. Poor solubility
and bioavailability are the main factors that limit its clinical application. Various structural …

In vitro synergistic effect of hesperidin and doxorubicin downregulates epithelial-mesenchymal transition in highly metastatic breast cancer cells

ND Amalina, IA Salsabila, UM Zulfin, RI Jenie… - Journal of the Egyptian …, 2023 - Springer
Background We previously reported that in highly metastatic breast cancer cells, doxorubicin
(DOX) at non-toxic concentrations promoted cell migration and invasion. Hesperidin (30, 5, 9 …

MAT as a promising therapeutic strategy against triple-negative breast cancer via inhibiting PI3K/AKT pathway

S Wei, Y Zhang, X Ma, Y Yao, Q Zhou, W Zhang… - Scientific Reports, 2023 - nature.com
Triple-negative breast cancer (TNBC), a highly aggressive and heterogeneous subtype of
breast cancer, lacks effective treatment options. Sophora flavescens Aiton, a Chinese …

[HTML][HTML] Chemoprevention curcumin analog 1.1 promotes metaphase arrest and enhances intracellular reactive oxygen species levels on TNBC MDA-MB-231 and …

D Novitasari, RI Jenie, J Kato… - Research in …, 2023 - journals.lww.com
Background and purpose: Previous studies highlighted that chemoprevention curcumin
analog-1.1 (CCA-1.1) demonstrated an antitumor effect on breast, leukemia, and colorectal …

Identification of potential targets of the curcumin analog CCA-1.1 for glioblastoma treatment: integrated computational analysis and in vitro study

A Hermawan, F Wulandari, N Hanif, RY Utomo… - Scientific Reports, 2022 - nature.com
The treatment of glioblastoma multiforme (GBM) is challenging owing to its localization in the
brain, the limited capacity of brain cells to repair, resistance to conventional therapy, and its …

Virtual screening of potential inhibitor against breast cancer-causing estrogen receptor alpha (ERα): molecular docking and dynamic simulations

S Muhammad, A Saba, RA Khera… - Molecular …, 2022 - Taylor & Francis
Breast cancer (Bca) causes the highest rate of mortality in females owing to the out-of-
control cell division in breast cells. In this work, we perform an in-silico screening based on …

Pentagamavunone-1 inhibits aggressive breast cancer cell proliferation through mitotic catastrophe and ROS-mediated activities: in vitro and in vivo studies

D Novitasari, I Nakamae, RI Jenie… - Saudi Pharmaceutical …, 2024 - Elsevier
Abstract Pentagamavunone-1 (PGV-1), an analog of curcumin, has been studied for its
cytotoxic effects in 4T1, MCF7, MCF7/HER2, and T47D breast cancer cells. Its …

[HTML][HTML] Transcriptomics analyses reveal the effects of Pentagamaboronon-0-ol on PI3K/Akt and cell cycle of HER2+ breast cancer cells

A Hermawan, F Wulandari, RY Utomo… - Saudi Pharmaceutical …, 2023 - Elsevier
Introduction Monoclonal antibodies and targeted therapies against HER2+ breast cancer
has improved overall and disease-free survival in patients; however, encountering drug …

Bioinformatic and molecular interaction studies uncover that CCA-1.1 and PGV-1 differentially target mitotic regulatory protein and have a synergistic effect against …

E Meiyanto, D Novitasari, RY Utomo… - Indonesian Journal of …, 2022 - journal.ugm.ac.id
Abstract Numerous studies demonstrated CCA-1.1, the modified compound from PGV-1,
inhibits tumor cells growth in breast and colorectal cancer. This time, we used bioinformatics …