Challenge and countermeasures for EGFR targeted therapy in non-small cell lung cancer

X Tian, T Gu, MH Lee, Z Dong - … et Biophysica Acta (BBA)-Reviews on …, 2022 - Elsevier
Lung cancer causes the highest mortality compared to other cancers in the world according
to the latest WHO reports. Non-small cell lung cancer (NSCLC) contributes about 85% of …

Safety and tolerability of epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors in oncology

RR Shah, DR Shah - Drug safety, 2019 - Springer
Tyrosine kinase inhibitors (TKIs) that target epidermal growth factor receptor (EGFR) have
dramatically improved progression-free survival in non-small-cell lung cancer (NSCLC) …

Overview of the multifaceted resistances toward EGFR-TKIs and new chemotherapeutic strategies in non-small cell lung cancer

RD Keflee, KH Leong, S Ogawa, J Bignon… - Biochemical …, 2022 - Elsevier
The role of epidermal growth factor receptor (EGFR) in non-small cell lung cancer (NSCLC)
has been vastly studied over the last decade. This has led to the rapid development of many …

Afatinib helped overcome subsequent resistance to osimertinib in a patient with NSCLC having leptomeningeal metastasis baring acquired EGFR L718Q mutation: a …

J Liu, B Jin, H Su, X Qu, Y Liu - BMC cancer, 2019 - Springer
Background The epidermal growth factor receptor (EGFR)-mutated advanced non-small-cell
lung cancer has been successfully treated with tyrosine kinase inhibitors (TKIs). Acquired …

Comparison of resistance spectra after first and second line osimertinib treatment detected by liquid biopsy

B Jóri, S Schatz, L Kaller, B Kah, J Roeper… - Cancers, 2021 - mdpi.com
Simple Summary Since the recent approval of osimertinib, a third generation tyrosine kinase
inhibitor (TKI) targeting EGFR in non-small cell lung cancer (NSCLC), tracing the resistance …

Metabolic radiogenomics in lung cancer: associations between FDG PET image features and oncogenic signaling pathway alterations

G Kim, J Kim, H Cha, WY Park, JS Ahn, MJ Ahn… - Scientific reports, 2020 - nature.com
This study investigated the associations between image features extracted from tumor 18F-
fluorodeoxyglucose (FDG) uptake and genetic alterations in patients with lung cancer. A …

Case report: dacomitinib may not benefit patients who develop rare compound mutations after later-line osimertinib treatment

HS Li, GJ Yang, Y Wang - Frontiers in oncology, 2021 - frontiersin.org
The acquired EGFR C797X mutation has been identified as the most notable resistance to
osimertinib, and novel secondary mutations of EGFR L718 and L792 residues have also …

CRISPER/CAS system, a novel tool of targeted therapy of drug-resistant lung cancer

VA Kordkheyli, M Rashidi, Y Shokri… - Advanced …, 2021 - pmc.ncbi.nlm.nih.gov
Lung cancer (LC) is the most common cause of cancer-related death worldwide. Patients
with LC are usually diagnosed at advanced phases. Five-year survival rate in LC patients is …

Comparative analysis of batch correction methods for FDG PET/CT using metabolic radiogenomic data of lung cancer patients

H Lee, S Seo, S Won, WY Park, JY Choi, KH Lee… - Scientific Reports, 2023 - nature.com
In radiomics research, the issue of different instruments being used is significant. In this
study, we compared three correction methods to reduce the batch effects in radiogenomic …

Structure Defines Function: Clinically Relevant Mutations in ErbB Kinases: Miniperspective

J Niggenaber, J Hardick, J Lategahn… - Journal of Medicinal …, 2019 - ACS Publications
The ErbB receptor tyrosine kinase family members EGFR (epidermal growth factor receptor)
and Her2 are among the prominent mutated oncogenic drivers of non-small cell lung cancer …