The bioactivity of thiazolidin-4-ones: A short review of the most recent studies
D Mech, A Kurowska, N Trotsko - International Journal of Molecular …, 2021 - mdpi.com
Thiazolidin-4-ones is an important heterocyclic ring system of a pharmacophore and a
privileged scaffold in medicinal chemistry. This review is focused on the latest scientific …
privileged scaffold in medicinal chemistry. This review is focused on the latest scientific …
[PDF][PDF] Substituted pyrimidine-sulfonamide derivatives: Computational, synthesis, characterization, anti-bacterial, MTT and molecular docking assessment
M Arshad, V Matiychuk - Biointerface Res. Appl. Chem, 2022 - biointerfaceresearch.com
A series of 4-[2-Amino-6-(3, 4, 5-substituted-phenyl) pyrimidin-4-yl] benzenesulfonamide (1-
6) was designed and assessed for bioactivity score and physicochemical analysis. All …
6) was designed and assessed for bioactivity score and physicochemical analysis. All …
Synthesis, Characterization, Antimicrobial, and Molecular Docking Studies of Thiazolidin-4-one Derivatives fused with Indole and Pyrimidine Moieties
A series of fifteen 2-substituted-3-(4-(pyridin-2-yl)-6-(1 H-pyrrolo [2, 3-b] pyridin-4-yl)
pyrimidin-2-yl) thiazolidin-4-one, was prepared and characterized using analytical …
pyrimidin-2-yl) thiazolidin-4-one, was prepared and characterized using analytical …
Synthesis, Characterization, Biological, and Molecular Docking Studies of (Z)-N-Substituted-4-(Pyridin-2-yl)-6-(1H-Pyrrolo[2,3-b]Pyridin-4-yl)Pyrimidin-2-Amine
M Arshad, MS Akhter - Russian Journal of Bioorganic Chemistry, 2022 - Springer
A series of fifteen (Z)-N-substituted-4-(pyridin-2-yl)-6-(1 H-pyrrolo [2, 3-b] pyridin-4-yl)
pyrimidin-2-amine, was designed, screened computationally and synthesized. Structures of …
pyrimidin-2-amine, was designed, screened computationally and synthesized. Structures of …
Design, Synthesis, Characterization, Antimicrobial, Anticancer Studies of Novel Thiazolidin-4-one Derivatives
Objective: Microbial infections and the cancer are the biggest health concerns now days. It
has been reported that 19.3 million new cancer cases and approximately 10 million deaths …
has been reported that 19.3 million new cancer cases and approximately 10 million deaths …
Discovery of Repurposable Drugs in the Combination Therapy of Breast Cancer: A Virtual Drug Screening Study
E Kırmızıay, R Demir, C Öğütçü… - Turkish Computational …, 2024 - dergipark.org.tr
Cathepsin D (Cat D) is a lysosomal aspartic acid protease encoded by CTSD gene and has
significant biological roles such as degradation of extracellular and intracellular proteins …
significant biological roles such as degradation of extracellular and intracellular proteins …