Highly reactive 4-membered ring nitrogen-containing heterocycles: synthesis and properties

B Alcaide, P Almendros, C Arangocillo - 2010 - digital.csic.es
4-Membered nitrogen-containing heterocycles, such as β-lactams (ie, 2-azetidinones) and
azetidines, are useful substrates in organic chemistry for the design and preparation of …

Ring expansions of activated aziridines and azetidines

MK Ghorai, A Bhattacharyya, S Das… - Synthesis of 4-to 7 …, 2016 - Springer
Facile construction of small and normal-sized, or more precisely, four to seven-membered
aza-heterocyclic ring systems is always a challenging yet rewarding task for the synthetic …

BF3·OEt2-Mediated Highly Regioselective SN2-Type Ring-Opening of N-Activated Aziridines and N-Activated Azetidines by Tetraalkylammonium Halides

MK Ghorai, A Kumar, DP Tiwari - The Journal of organic chemistry, 2010 - ACS Publications
A highly regioselective Lewis acid-mediated SN2-type ring-opening of N-sulfonylaziridines
and azetidines with tetraalkylammonium halides in CH2Cl2 solution to afford 1, 2-and 1, 3 …

[PDF][PDF] Preparation and synthetic applications of azetidines

TM Bott, FG West - Heterocycles, 2012 - triggered.stanford.clockss.org
Azetidines (four-membered saturated nitrogen heterocycles) are found in a diverse range of
natural products, and also serve as valuable building blocks for other structural classes. The …

Syntheses of chiral β-and γ-amino ethers, morpholines, and their homologues via nucleophilic ring-opening of chiral activated aziridines and azetidines

MK Ghorai, D Shukla… - The Journal of Organic …, 2012 - ACS Publications
Lewis acid catalyzed quaternary ammonium salt mediated highly regioselective ring-
opening of chiral activated aziridines and azetidines with alcohols to nonracemic β-and γ …

Lewis acid catalyzed highly stereoselective domino-ring-opening cyclization of activated aziridines with enolates: synthesis of functionalized chiral γ-lactams

MK Ghorai, DP Tiwari - The Journal of Organic Chemistry, 2010 - ACS Publications
A highly enantio-and diastereoselective Lewis acid catalyzed SN2-type ring opening
followed by cyclization of aziridines with active methylene carbon nucleophiles to …

Stereospecific synthesis of 1, 4, 5, 6-tetrahydropyrimidines via domino ring-opening cyclization of activated aziridines with α-acidic isocyanides

A Bhattacharyya, CK Shahi, S Pradhan… - Organic letters, 2018 - ACS Publications
An expeditious synthetic route to access structurally diverse 1, 4, 5, 6-tetrahydropyrimidines
via domino ring-opening cyclization of activated aziridines with α-acidic isocyanides has …

Enantioselective Syntheses of Morpholines and Their Homologues via SN2-Type Ring Opening of Aziridines and Azetidines with Haloalcohols

MK Ghorai, D Shukla, K Das - The Journal of Organic Chemistry, 2009 - ACS Publications
A highly regio-and stereoselective strategy for the syntheses in high yield and
enantioselectivity of a variety of substituted nonracemic morpholines and their homologues …

Synthetic route to chiral tetrahydroquinoxalines via ring-opening of activated aziridines

MK Ghorai, AK Sahoo, S Kumar - Organic Letters, 2011 - ACS Publications
A highly regio-and stereoselective route for the synthesis of racemic and nonracemic
tetrahydroquinoxalines via the SN2-type ring-opening of activated aziridines with 2 …

Ring opening/C–N cyclization of activated aziridines with carbon nucleophiles: highly diastereo-and enantioselective synthesis of tetrahydroquinolines

MK Ghorai, Y Nanaji, AK Yadav - Organic Letters, 2011 - ACS Publications
A simple strategy for the synthesis of substituted tetrahydroquinolines through regio-and
stereoselective ring opening of N-tosyl aziridines with carbon nucleophiles generated from 2 …