Thiazole ring—A biologically active scaffold
A Petrou, M Fesatidou, A Geronikaki - Molecules, 2021 - mdpi.com
Background: Thiazole is a good pharmacophore nucleus due to its various pharmaceutical
applications. Its derivatives have a wide range of biological activities such as antioxidant …
applications. Its derivatives have a wide range of biological activities such as antioxidant …
Development and therapeutic potential of 2-aminothiazole derivatives in anticancer drug discovery
SR Alizadeh, SM Hashemi - Medicinal Chemistry Research, 2021 - Springer
Currently, the development of anticancer drug resistance is significantly restricted the clinical
efficacy of the most commonly prescribed anticancer drug. Malignant disease is widely …
efficacy of the most commonly prescribed anticancer drug. Malignant disease is widely …
A retrospect on antimicrobial potential of thiazole scaffold
Due to its appreciable diversity in biological actions, thiazole and its substituted
components, a significant class of heterocyclic compounds has developed as an influential …
components, a significant class of heterocyclic compounds has developed as an influential …
Anticancer potential of thiazole derivatives: a retrospective review
S Jain, S Pattnaik, K Pathak, S Kumar… - Mini reviews in …, 2018 - ingentaconnect.com
This review brings forth the potential of thiazole derivatives for their anticancer activities. The
emphasis is placed on the structural diversity of thiazole derivatives, responsible for their …
emphasis is placed on the structural diversity of thiazole derivatives, responsible for their …
[PDF][PDF] Antibacterial activity of thiazole and its derivatives
Thiazoles are one of the most intensively scrutinized classes of 5-membered aromatic
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …
heterocycles. Many natural and synthesized thiazole and its derivatives showed significant …
Review on synthetic chemistry and antibacterial importance of thiazole derivatives
A Kashyap, N Adhikari, A Das, A Shakya… - Current drug …, 2018 - ingentaconnect.com
Background: Thiazole is one of the leading heterocyclic five-member ring compounds that
contain nitrogen and sulphur atom. Many natural and/or synthetic compounds contain …
contain nitrogen and sulphur atom. Many natural and/or synthetic compounds contain …
Heterocycle compounds with antimicrobial activity
M Fesatidou, A Petrou, G Athina - Current pharmaceutical …, 2020 - ingentaconnect.com
Background: Bacterial infections are a growing problem worldwide causing morbidity and
mortality mainly in developing countries. Moreover, the increased number of …
mortality mainly in developing countries. Moreover, the increased number of …
2, 4-Disubstituted thiazoles as multitargated bioactive molecules
Thiazoles are important heterocyclics exhibiting boundaryless biological activities, such as
antibacterial, antifungal, anti-inflammatory, antitumor, antitubercular, antidiabetic, antiviral …
antibacterial, antifungal, anti-inflammatory, antitumor, antitubercular, antidiabetic, antiviral …
Synthesis, in silico and biological studies of thiazolyl-2h-chromen-2-one derivatives as potent antitubercular agents
BS Jadhav, RS Yamgar, RS Kenny… - … -Aided Drug Design, 2020 - ingentaconnect.com
Background: A series of new six thiazolyl-2-amine-based Schiff base derivatives (4a-4f)
were synthesized by a sequential multistep reaction starting with Salicylaldehyde. Methods …
were synthesized by a sequential multistep reaction starting with Salicylaldehyde. Methods …
[HTML][HTML] Quorum sensing inhibitors: curbing pathogenic infections through inhibition of bacterial communication
Currently, most of the developed and developing countries are facing the problem of
infectious diseases. The genius way of an exaggerated application of antibiotics led the …
infectious diseases. The genius way of an exaggerated application of antibiotics led the …