Current strategies in development of new chromone derivatives with diversified pharmacological activities: A review
NA Mohsin, M Irfan, S Hassan, U Saleem - Pharmaceutical chemistry …, 2020 - Springer
Chromone derivatives possess a spectrum of biological activities. Chromone has been
recognized as a privileged structure for new drug invention and development. Substitution …
recognized as a privileged structure for new drug invention and development. Substitution …
Ramachary-Bressy-Wang [3+ 2] cycloaddition reaction: Synthesis of fully decorated 1, 2, 3-triazoles as potent anticancer and EGFR inhibitors
M Kumar, SK Nukala, NS Thirukovela… - Journal of Molecular …, 2022 - Elsevier
A general strategy was developed for the synthesis of new fully decorated 1, 2, 3-triazoles
(5a-m & 6a-e) containing coumarine and sulfonyl-benzimidazole from 3-(2-((1-methyl-1H …
(5a-m & 6a-e) containing coumarine and sulfonyl-benzimidazole from 3-(2-((1-methyl-1H …
Design, synthesis and biological evaluation of novel 1, 2, 3-triazole-based xanthine derivatives as DPP-4 inhibitors
Inhibitors of dipeptidyl peptidase-4 (DPP4) have been shown to be effective treatments for
type 2 diabetes. A series of novel 1, 2, 3-triazole based xanthine derivatives were designed …
type 2 diabetes. A series of novel 1, 2, 3-triazole based xanthine derivatives were designed …
Microwave-assisted Cu-catalyzed C–C bond formation: one-pot synthesis of fully substituted 1, 2, 3-triazoles using nonsymmetrical iodoalkynes and their biological …
S Narsimha, KS Battula, YN Reddy… - Chemistry of Heterocyclic …, 2018 - Springer
A copper-catalyzed one-pot synthesis of fused benzothiazino [1, 2, 3] triazolo [4, 5-c]
quinolinone derivatives from 1-iodoalkynes with different aryl azides via an in situ generated …
quinolinone derivatives from 1-iodoalkynes with different aryl azides via an in situ generated …
Synthesis, characterization and biological evaluation of 7-substituted-4-((1-aryl-1H-1, 2, 3-triazol-4-yl) methyl)-2H-benzo [b][1, 4] oxazin-3 (4H)-ones as anticancer …
VR Nagavelli, SK Nukala, S Narsimha… - Medicinal Chemistry …, 2016 - Springer
Abstract A series of novel 1, 2, 3-triazole-2H-benzo [b][1, 4] oxazin-3 (4H)-ones (4a–4k and
5a–5g) were designed, synthesized and screened for their anticancer activity against MCF-7 …
5a–5g) were designed, synthesized and screened for their anticancer activity against MCF-7 …
One-pot synthesis of novel 1, 2, 3-triazole-pyrimido [4, 5-c] isoquinoline hybrids and evaluation of their antioxidant activity
S Narsimha, KS Battula, VR Nagavelli - Synthetic Communications, 2018 - Taylor & Francis
ABSTRACT A series of novel pyrimido [4, 5-c] isoquinolines (3a–3h) and 1, 2, 3-triazole-
coupled pyrimido [4, 5-c] isoquinolines (4a–4h) were synthesized in good to excellent yields …
coupled pyrimido [4, 5-c] isoquinolines (4a–4h) were synthesized in good to excellent yields …
One-pot synthesis of sulfonyl-1H-1,2,3-triazolyl-thiomorpholine 1,1-dioxide derivatives and evaluation of their biological activity
R Sreerama, VR N, S Narsimha - Phosphorus, Sulfur, and Silicon …, 2020 - Taylor & Francis
A one-pot procedure for the synthesis of novel 1, 2, 3-triazole derivatives (5a–5l) in good
yields (63 to 77%) using different sulfonic acids and 4-(prop-2-yn-1-yl) thiomorpholine 1, 1 …
yields (63 to 77%) using different sulfonic acids and 4-(prop-2-yn-1-yl) thiomorpholine 1, 1 …
[HTML][HTML] Synthesis, anticancer and antibacterial evaluation of novel (isopropylidene) uridine-[1, 2, 3] triazole hybrids
R kumar Thatipamula, S Narsimha, K Battula… - Journal of Saudi …, 2017 - Elsevier
A series of novel (isopropylidene) uridine-[1, 2, 3] triazole hybrids (3a–3n) were efficiently
synthesized via the copper-catalyzed azide–alkyne cycloaddition (CuAAC) from N-propargyl …
synthesized via the copper-catalyzed azide–alkyne cycloaddition (CuAAC) from N-propargyl …
Synthesis and biological evaluation of novel thiomorpholine 1, 1‐dioxide derived 1, 2, 3‐triazole hybrids as potential anticancer agents
KS Battula, S Narsimha, RK Thatipamula… - …, 2017 - Wiley Online Library
In this report, we describe the synthesis and biological evaluation of a new series of (4‐((1‐
(aryl)‐1H‐1, 2, 3‐triazol‐4‐yl) methoxy) phenyl)(1, 1‐dioxidothiomorpholino) methanone …
(aryl)‐1H‐1, 2, 3‐triazol‐4‐yl) methoxy) phenyl)(1, 1‐dioxidothiomorpholino) methanone …
Synthesis and Biological Evaluation of (N‐(3‐methoxyphenyl)‐4‐((aryl‐1H‐1,2,3‐triazol‐4‐yl)methyl)thiomorpholine‐2‐carboxamide 1,1‐Dioxide Hybrids as …
KS Battula, S Narsimha, RK Thatipamula… - …, 2017 - Wiley Online Library
A series of new thirteen N‐(3‐Methoxyphenyl) thiomorpholine‐2‐carboxamide 1, 1‐dioxide
derived 1, 4‐disubtituted 1, 2, 3‐triazole hybrids (7 a‐7 m) were synthesized by Cu (I) …
derived 1, 4‐disubtituted 1, 2, 3‐triazole hybrids (7 a‐7 m) were synthesized by Cu (I) …