Abstract 140 Years ago Adolf von Baeyer proposed the structure of a heteroaromatic
compound which revolutionized organic and medical chemistry: indole. After more than a …

Copper nanoparticles have been explored as a new class of heterogeneous catalyst in
various chemical transformations. This review surveys the most useful organic …

The direct and site‐selective transition metal‐catalysed N1‐, C2‐or C3‐arylations of indoles
have been the subject of almost continuous improvements since their discovery in early …

Abstract Vor 140 Jahren schlug Adolf von Baeyer die Struktur für eine heteroaromatische
Verbindung vor, die die organische und medizinische Chemie nachhaltig veränderte: Indol …

The N-arylation of indoles, including a variety of substituted ones, has been carried out
using bulky, electron-rich phosphines as the supporting ligand in combination with Pd2 …

This article describes the expected phenotypic behavior of all types of ligands in
constitutively active receptor systems and, in particular, the molecular mechanisms of …

(Chemical Equation Presented) A single tandem operation allows rapid access to a variety
of substituted N-functionalized indoles. The nitrogen atom of the indole nucleus is …

Melatonin had previously been shown to reduce up to four 2, 2 '‐azino‐bis‐(3‐
ethylbenzthiazoline‐6‐sulfonic acid) cation radicals (ABTS•+) via a scavenger cascade …

Lufotrelvir was designed as a first in class 3CL protease inhibitor to treat COVID-19.
Development of lufotrelvir was challenged by its relatively poor stability due to its propensity …

Melatonin MT1 and MT2 receptor ligands have been vigorously explored for the last 4
decades. Inspection of approximately 80 publications in the field revealed that most …