Comprehensive overview of carboxamide derivatives as succinate dehydrogenase inhibitors

B Luo, Y Ning - Journal of Agricultural and Food Chemistry, 2022 - ACS Publications
Up to now, a total of 24 succinate dehydrogenase inhibitors (SDHIs) fungicides have been
commercialized, and SDHIs fungicides were also one of the most active fungicides …

Recent advances in indazole-containing derivatives: synthesis and biological perspectives

SG Zhang, CG Liang, WH Zhang - Molecules, 2018 - mdpi.com
Indazole-containing derivatives represent one of the most important heterocycles in drug
molecules. Diversely substituted indazole derivatives bear a variety of functional groups and …

A review on synthetic strategy, molecular pharmacology of indazole derivatives, and their future perspective

S Mal, U Malik, M Mahapatra, A Mishra… - Drug Development …, 2022 - Wiley Online Library
With different nitrogen‐containing heterocyclic moieties, Indazoles earn one of the places
among the top investigated molecules in medicinal research. Indazole, an important fused …

Morpholine derivatives in agrochemical discovery and development

X Tang, L Lei, A Liao, W Sun, J Zhang… - Journal of Agricultural …, 2023 - ACS Publications
Derivatives of morpholine are biologically active organic compounds with special structures
discovered in multiple drugs. As a result of the terminal pharmacophore of action and …

Design, synthesis, DFT study and antifungal activity of pyrazolecarboxamide derivatives

JX Mu, YX Shi, MY Yang, ZH Sun, XH Liu, BJ Li… - Molecules, 2016 - mdpi.com
A series of novel pyrazole amide derivatives were designed and synthesized by multi-step
reactions from phenylhydrazine and ethyl 3-oxobutanoate as starting materials, and their …

Synthesis, Antifungal Activity and Structure-Activity Relationships of Novel 3-(Difluoromethyl)-1-methyl-1H-pyrazole-4-carboxylic Acid Amides

S Du, Z Tian, D Yang, X Li, H Li, C Jia, C Che, M Wang… - Molecules, 2015 - mdpi.com
A series of novel 3-(difluoromethyl)-1-methyl-1 H-pyrazole-4-carboxylic acid amides were
synthesized and their activities were tested against seven phytopathogenic fungi by an in …

44. Antioxidant, antimicrobial activity and phytochemical analysis of the seeds extract of Cucumis sativus Linn

HA Begum, F Asad, A Sadiq, S Mulk, K Ali - Pure and Applied Biology …, 2019 - thepab.org
The prehistoric interaction of plants and human is being strengthened by the remarkable use
of plants as remedy against diseases. Cucumis sativus L. is extensively cultivated globally …

Molecular dynamics and 3D-QSAR studies on indazole derivatives as HIF-1α inhibitors

Y Singh, KS Sanjay, P Kumar, S Singh… - Journal of Biomolecular …, 2023 - Taylor & Francis
Hypoxia-inducible factor (HIF) is a transcriptional factor which plays a crucial role in tumour
metastasis thereby responsible for development of various forms of cancers. Indazole …

1, 2, 4-Oxadiazole-based bio-isosteres of benzamides: Synthesis, biological activity and toxicity to zebrafish embryo

S Yang, CL Ren, TY Ma, WQ Zou, L Dai… - International Journal of …, 2021 - mdpi.com
To discover new compounds with broad spectrum and high activity, we designed a series of
novel benzamides containing 1, 2, 4-oxadiazole moiety by bioisosterism, and 28 …

Design, synthesis, and antifungal activity of novel aryl-1, 2, 3-triazole-β-carboline hybrids

XY Huo, L Guo, XF Chen, YT Zhou, J Zhang, XQ Han… - Molecules, 2018 - mdpi.com
The copper catalytic azide and terminal alkyne cycloaddition reaction, namely “click
chemistry”, gives a new and convenient way to create l, 4-disubstitutd-l, 2, 3-triazoles. In this …