Review of synthesis of 1, 3, 4-oxadiazole derivatives
KD Patel, SM Prajapati, SN Panchal… - Synthetic …, 2014 - Taylor & Francis
Oxadiazole nucleus shows a broad spectrum of pharmaceutical applications. Thus, in recent
years scientists have developed various new methods for the synthesis of its derivatives …
years scientists have developed various new methods for the synthesis of its derivatives …
Synthesis and antifungal activities of 5-(3, 4, 5-trimethoxyphenyl)-2-sulfonyl-1, 3, 4-thiadiazole and 5-(3, 4, 5-trimethoxyphenyl)-2-sulfonyl-1, 3, 4-oxadiazole …
CJ Chen, BA Song, S Yang, GF Xu, PS Bhadury… - Bioorganic & medicinal …, 2007 - Elsevier
Starting from the key intermediate 5-(3, 4, 5-trimethoxyphenyl)-1, 3, 4-thiadiazole-2-thiol (4)
or the oxadiazole analogue (5), the title compounds 9 and 10 are synthesized by a two-step …
or the oxadiazole analogue (5), the title compounds 9 and 10 are synthesized by a two-step …
Synthesis, structure, and bioactivity of N′-substituted benzylidene-3, 4, 5-trimethoxybenzohydrazide and 3-acetyl-2-substituted phenyl-5-(3, 4, 5-trimethoxyphenyl)-2 …
L Jin, J Chen, B Song, Z Chen, S Yang, Q Li… - Bioorganic & medicinal …, 2006 - Elsevier
Some 3-acetyl-2-substituted phenyl-5-(3, 4, 5-trimethoxyphenyl)-2, 3-dihydro-1, 3, 4-
oxadiazole derivatives were synthesized by cyclization reaction of N′-substituted …
oxadiazole derivatives were synthesized by cyclization reaction of N′-substituted …
[HTML][HTML] Biochemical evaluation of a series of synthetic chalcone and hydrazide derivatives as novel inhibitors of cruzain from Trypanosoma cruzi
DM Borchhardt, A Mascarello, LD Chiaradia… - Journal of the Brazilian …, 2010 - SciELO Brasil
Chagas' disease, a parasitic infection widely distributed throughout Latin America, is a major
public health problem with devastating consequences in terms of human morbidity and …
public health problem with devastating consequences in terms of human morbidity and …
Electrocyclization of semicarbazone; A novel route of green synthesis of 2, 5-disubstituted-1, 3, 4-oxadiazoles
B Lotfi, B Mustafa, B Leila, M Salima - International Journal of …, 2011 - Elsevier
The anodic oxidation of a number of arylsemicarbazides derivatives (I) has been examined
in acetonitril containing lithium perchlorate (LiClO4) as a supporting electrolyte (20g/l). The …
in acetonitril containing lithium perchlorate (LiClO4) as a supporting electrolyte (20g/l). The …
[PDF][PDF] Synthesis and biological screening of some new substituted-3H-quinazolin-4-one analogs as antimicrobial agents
MA Al-Omar, SG Abdel Hamide… - Saudi pharmaceutical …, 2005 - academia.edu
A new series of substituted 3-benzyl-3H-quinazolin-4-one analogs was prepared and
screened for their antimicrobial activity. Compound 2-(3-nitro-2-pyridyl) thio-3-benzyl-6 …
screened for their antimicrobial activity. Compound 2-(3-nitro-2-pyridyl) thio-3-benzyl-6 …
An expeditious and one-pot synthesis of unsymmetrical 2, 5-disubstituted-1, 3, 4-oxadiazoles under microwave irradiation and solvent-free conditions
N Montazeri, K Rad-Moghadam - Chinese Chemical Letters, 2008 - Elsevier
A one-pot synthesis of some unsymmetrical 2, 5-disubstituted-1, 3, 4-oxadiazoles via
cyclocondensation of benzoylhydrazines with orthoesters under solvent-free and microwave …
cyclocondensation of benzoylhydrazines with orthoesters under solvent-free and microwave …
[PDF][PDF] Synthesis and biological screening of some new substituted 2-mercapto-4 (3H) quinazolinone analogues as anticonvulsant agents
Epilepsy is a very common disorder, characterized by seizures, which takes various form
and result from episodic neuronal discharges. Current antiepileptic drugs are effective in …
and result from episodic neuronal discharges. Current antiepileptic drugs are effective in …
1, 3, 4-Oxadiazole formation; a novel solid support strategy
JP Kilburn, J Lau, RCF Jones - Tetrahedron Letters, 2001 - Elsevier
A new approach to the synthesis of 1, 3, 4-oxadiazoles on solid support is described. Resin
bound 1-acyl thiosemicarbazides were treated with a variety of dehydrating agents at …
bound 1-acyl thiosemicarbazides were treated with a variety of dehydrating agents at …
(2-Arylhydrazonomethyl)-substituted xanthones as antimycotics: synthesis and fungistatic activity against Candida species
S Moreau, M Varache-Lembège, S Larrouture… - European journal of …, 2002 - Elsevier
A series of arylhydrazones derived from various 6, 8-diacetoxy-or 6, 8-dihydroxy-9-oxo-9H-
xanthene carboxaldehydes were synthesized and evaluated for their in vitro antifungal …
xanthene carboxaldehydes were synthesized and evaluated for their in vitro antifungal …