Novel combinations
F Burkamp, P Hansen - US Patent App. 12/749,888, 2010 - Google Patents
The invention provides a pharmaceutical product comprising, in combination,(1) a named
glucocorticosteroid receptor agonist and (2) a B adrenoreceptoragonist, a dual 32 adreno …
glucocorticosteroid receptor agonist and (2) a B adrenoreceptoragonist, a dual 32 adreno …
Novel compounds
F Burkamp, P Hansen - US Patent App. 12/749,919, 2010 - Google Patents
0002 The present invention relates to compounds having glucocorticosteroid receptor
agonist activity, processes for their preparation, pharmaceutical compositions containing …
agonist activity, processes for their preparation, pharmaceutical compositions containing …
Combination steroid and glucocorticoid receptor antagonist therapy
J Belanoff, P Lockey - US Patent 8,829,024, 2014 - Google Patents
The present invention provides compositions of an anti-in flammatory glucocorticosteroid
and a glucocorticoid recep tor (GR) modulator useful for inhibiting glucocorticoid receptor …
and a glucocorticoid recep tor (GR) modulator useful for inhibiting glucocorticoid receptor …
Novel amide compounds
F Burkamp, B Gabos, S Ivanova… - US Patent App. 12 …, 2010 - Google Patents
0002 The present invention relates to compounds having glucocorticosteroid receptor
agonist activity, processes for their preparation, pharmaceutical compositions containing …
agonist activity, processes for their preparation, pharmaceutical compositions containing …
Novel Amide Compounds
F Burkamp, B Gabos, S Ivanova… - US Patent App. 13 …, 2013 - Google Patents
0002 The present invention relates to compounds having glucocorticosteroid receptor
agonist activity, processes for their preparation, pharmaceutical compositions containing …
agonist activity, processes for their preparation, pharmaceutical compositions containing …
Highly potent glucocorticoids
US9975918B2 - Highly potent glucocorticoids - Google Patents US9975918B2 - Highly potent
glucocorticoids - Google Patents Highly potent glucocorticoids Download PDF Info Publication …
glucocorticoids - Google Patents Highly potent glucocorticoids Download PDF Info Publication …
Medicament for treating peripheral neuropathies
HL Yu - US Patent 9,526,729, 2016 - Google Patents
0 [1*] C (N) C (= O) OCCOCN1C= NC2= C1N= C (N) N= C2O Chemical compound [1*] C (N)
C (= O) OCCOCN1C= NC2= C1N= C (N) N= C2O 0.000 description 2AHFHDYBIPSFVCP …
C (= O) OCCOCN1C= NC2= C1N= C (N) N= C2O 0.000 description 2AHFHDYBIPSFVCP …
Structures and mechanism for the design of highly potent glucocorticoids
Adcock, IM, et al.(1999) Ligand-induced differentiation of glucocorticoid receptor (GR) trans-
repression and transactivation: preferential targetting of NF-kappaB and lack of I-kappaB …
repression and transactivation: preferential targetting of NF-kappaB and lack of I-kappaB …