In recent years, transition‐metal‐catalyzed C− H activation has become a key strategy in the
field of organic synthesis. Rhodium complexes are widely used as catalysts in a variety of …

Sulfonamide derivatives are frequently seen structural motifs in medicinal chemistry. Almost
a century after Gerhard Domagk's pioneering work leading to the first sulfonamide antibiotic …

Sulfoximines have been largely disregarded in medicinal chemistry for a long time.
However, recently, they have risen to the apparent level of stardom on the drug discovery …

sulfinamides, sulfonamides, and sulfonimidamides are in-demand motifs in medicinal
chemistry, yet methods for the synthesis of alkyl variants that start from simple, readily …

New methods for the general asymmetric synthesis of sulfonimidamides are of great interest
due to their applications in medicinal chemistry, agrochemical discovery, and academic …

Historically, sulfoximines, sulfondiimines and sulfonimidamides have been neglected
pharmacophores in drug discovery even though they offer very interesting properties. This …

Chiral sulfinyl compounds, sulfoxides, sulfoximines, sulfinamides, and other derivatives, play
an important role in asymmetric synthesis as versatile auxiliaries, ligands, and catalysts …

Achiral sulfur functional groups, such as sulfonamide, sulfone, thiol and thioether, are
common in drugs and natural products. By contrast, chiral sulfur functional groups are often …

Sulfur can form diverse S (IV) and S (VI) stereogenic centers, of which some have gained
significant attention recently due to their increasing use as pharmacophores in drug …

Extension of the medicinal chemistry toolbox is in the vital interest of drug designers.
However, the diffusion of an innovation can be a lengthy process. Along these lines, it took …