Polymers for Disrupting Protein–Protein Interactions: Where Are We and Where Should We Be?

SP Le, J Krishna, P Gupta, R Dutta, S Li… - …, 2024 - ACS Publications
Protein–protein interactions (PPIs) are central to the cellular signaling and regulatory
networks that underlie many physiological and pathophysiological processes. It is …

Exploring the potential of P-glycoprotein inhibitors in the targeted delivery of anti-cancer drugs: A comprehensive review

D Patel, N Sethi, P Patel, S Shah, K Patel - European Journal of …, 2024 - Elsevier
Due to the high prevalence of cancer, progress in the management of cancer is the need of
the hour. Most cancer patients develop chemotherapeutic drug resistance, and many remain …

Exploring the effects of pemetrexed on drug resistance mechanisms in human lung adenocarcinoma and its association with PGRMC1

SY Wu, EC Liao, YF Wen, YS Wang, H Meng… - Chemico-Biological …, 2024 - Elsevier
According to the 2022 cancer statistics of the World Health Organization, lung cancer ranks
among the top ten causes of death, with lung adenocarcinoma being the most prevalent …

Pharmaceutical prospects of pomegranate antioxidants in combating microbial infections

R Malkawi, B Jarwan, R Waleed… - International Journal of …, 2024 - Taylor & Francis
Pomegranates, which are renowned for their diverse bioactive phytochemicals with
antioxidant, anti-inflammatory, and antimicrobial properties, have garnered significant …

Interactions between multifunctional pharmaceutical excipients and efflux pump for optimal drug transport and bioavailability: An overview

VL Gaikwad, S Sen, PR Dhake - Journal of Drug Delivery Science and …, 2024 - Elsevier
Polymeric excipients ensure the site-specific delivery of the drug at the desired rate for a
specified duration to achieve better efficacy. Pharmaceutical excipients were supposed to be …

[HTML][HTML] Comparing antioxidant and cytoprotective effects: Quercetin glycoside vs. aglycone from Ephedra alata

E El Maaiden, N Ullah, A Ezzariai, A Mazar… - Phytomedicine Plus, 2024 - Elsevier
Background A wide range of chronic diseases is associated with ROS-mediated oxidative
stress. Quercetin glycoside (QG) is reported to be a powerful antioxidant with extremely high …

Design, Synthesis, Computational Study, and Biological Evaluation of Sulfonyl Tethered Piperazine Derivatives as Antimicrobial Agents

V Thopate, SA Dhawale, R Kawale, D Gaikwad… - …, 2024 - Wiley Online Library
Piperazine, a nitrogen‐containing heterocyclic compound, has potential in medical
chemistry due to its versatile structure and ease of modification. Therefore, researchers have …

Investigating natural inhibitors of Permeability-glycoprotein (P-gp) liver transporter via molecular docking simulation for Hepatocellular carcinoma therapy

A Dey, R Li, N Larzat, JB Idoipe, A Kati… - … Conference on Soft …, 2023 - Springer
Abstract Permeability-glycoprotein (P-gp), a dynamic efflux pump responsible for
transporting xenobiotics and drugs out of cells, is a contributor to multidrug resistance …

[PDF][PDF] Phytomedicine Plus

E El Maaiden, N Ullah, A Ezzariai, A Mazar, H Boukcim… - researchgate.net
Background: A wide range of chronic diseases is associated with ROS-mediated oxidative
stress. Quercetin glycoside (QG) is reported to be a powerful antioxidant with extremely high …