Calixarene-based phosphinic acids as inhibitors of protein tyrosine phosphatases
VM Buldenko, VV Trush, OL Kobzar… - Bioorganic & medicinal …, 2019 - Elsevier
In the present work, the derivatives of calix [4] arene, thiacalix [4] arene, and sulfonylcalix [4]
arene bearing four methylene (phenyl) phosphinic acid groups on the upper rim of the …
arene bearing four methylene (phenyl) phosphinic acid groups on the upper rim of the …
[HTML][HTML] Inhibition of glutathione S-transferases by photoactive calix [4] arene α-ketophosphonic acids
Calix [4] arenes bearing photoactive α-ketophosphonic acid groups at the upper rim of the
macrocycle were synthesized and evaluated as inhibitors of glutathione S-transferases …
macrocycle were synthesized and evaluated as inhibitors of glutathione S-transferases …
Phenylpyrazalopyrimidines as Tyrosine Kinase Inhibitors: Synthesis, Antiproliferative Activity, and Molecular Simulations
N 1-(α, β-Alkene)-substituted phenylpyrazolopyrimidine derivatives with acetyl and
functionalized phenyl groups at α-and β-positions, respectively, were synthesized by the …
functionalized phenyl groups at α-and β-positions, respectively, were synthesized by the …
Functional calixarenes for material and life science
R Rodik, S Cherenok, O Kalchenko… - Current Organic …, 2018 - ingentaconnect.com
Calix [n] arenes–are easily accessible three-dimensional macrocyclic compounds. Modified
calix [n] arenes capable with high selectivity recognize, bind in supramolecular complexes …
calix [n] arenes capable with high selectivity recognize, bind in supramolecular complexes …
Alkyl and aryl α-ketophosphonate derivatives as photoactive compounds targeting glutathione S-transferases
ОL Kobzar, YV Shulha, VM Buldenko… - … , Sulfur, and Silicon …, 2021 - Taylor & Francis
In this article, photoactive alkyl and aryl α-ketophosphonate derivatives were studied as
inhibitors of glutathione S-transferases (GSTs). The α-ketophosphonate monoesters were …
inhibitors of glutathione S-transferases (GSTs). The α-ketophosphonate monoesters were …
Calixarene derivatives for (nano) biotechnologies
This review summarizes the author's research in the field of bio-medical application of
modified calixarenes as well as their nano-associates. The paper includes results of design …
modified calixarenes as well as their nano-associates. The paper includes results of design …
Sulfonyl-bridged calix [4] arene as an inhibitor of protein tyrosine phosphatases
V Buldenko, O Kobzar, V Trush… - French-Ukrainian …, 2017 - kyivtoulouse.univ.kiev.ua
Previously, phosphonic acid derivatives of calix [4] arene and thiacalix [4] arene were found
to be potential inhibitors of protein tyrosine phosphatase 1B. In the present paper, the …
to be potential inhibitors of protein tyrosine phosphatase 1B. In the present paper, the …
Inhibition of glutathione S-transferases by calix [4] arene-based phosphinic acids
OL Kobzar, YV Shulha, VM Buldenko… - Ukrainica …, 2022 - bioorganica.com.ua
Abstract Calix [4] arene-, thiacalix [4] arene-and sulfonylcalix [4] arene-based derivatives
with upper rim phosphinic acid groups were studied as inhibitors of glutathione S …
with upper rim phosphinic acid groups were studied as inhibitors of glutathione S …
Functional calixarene nanostructures
VI Kalchenko - Theoretical and Experimental Chemistry, 2018 - Springer
The results of the author studies of functional calixarene nanostructures are summarized.
Calixarenes modified by various functional groups were created with receptor properties …
Calixarenes modified by various functional groups were created with receptor properties …
Biologically active calixarene phosphonic acids
Phosphorylated derivatives of organic compounds are known to be capable of inhibiting the
activities of enzymes and other proteins responsible for key metabolic pathways. In this …
activities of enzymes and other proteins responsible for key metabolic pathways. In this …