Biodegradable pH-responsive micelles loaded with 8-hydroxyquinoline glycoconjugates for Warburg effect based tumor targeting

A Domiński, M Krawczyk, T Konieczny… - European Journal of …, 2020 - Elsevier
Biodegradable triblock copolymer poly (ethylene glycol)-b-polycarbonate-b-oligo ([R]-3-
hydroxybutyrate) was prepared via metal-free ring-opening polymerization of ketal protected …

TLR7 endogenous ligands remodel glycolytic macrophages and trigger skin‐to‐joint crosstalk in psoriatic arthritis

K Van Raemdonck, S Umar… - European journal of …, 2021 - Wiley Online Library
Thirty percent of psoriasis patients develop psoriatic arthritis (PsA), nevertheless the
mechanism remains unknown. Endogenous GU‐rich miRNAs activate endosomal TLR7 that …

[PDF][PDF] The Impact of Proinflammatory Cytokines and Imiquimod on GLUT1 in HaCaT Keratinocytes–a Potential Anti-Psoriatic Therapeutic Target?

S Makuch, P Kupczyk, A Makarec… - Cell Physiol …, 2023 - articles.cellphysiolbiochem.com
Abstract Background/Aims: Glucose metabolism has been proven as an essential process
for proliferating keratinocytes, which highlights the importance of glucose transporter-1 …

In vitro and in vivo efficacy of a novel glucose–methotrexate conjugate in targeted cancer treatment

M Woźniak, G Pastuch-Gawołek, S Makuch… - International Journal of …, 2021 - mdpi.com
Methotrexate (MTX) is a commonly used antimetabolite, which inhibits folate and DNA
synthesis to be effective in the treatment of various malignancies. However, MTX therapy is …

Phytochemical investigation, structural elucidation, in silico study and anti-psoriatic activity of potent bioactive from Betula utilis

P Biswasroy, D Pradhan, DK Sahu, V Rai… - Journal of …, 2023 - Taylor & Francis
Psoriasis is a chronic autoimmune pathological condition characterized by hyperactivation
of proinflammatory cytokines (IL-6, TNF-α, IL-17, IL-23, etc.). Severe drug-associated …

Pithecellobium clypearia: Amelioration Effect on Imiquimod-Induced Psoriasis in Mice Based on a Tissue Metabonomic Analysis

Y Li, J Zong, W Ye, Y Fu, X Gu, W Pan… - Frontiers in …, 2021 - frontiersin.org
Pithecellobium clypearia Benth.(accepted name: Archidendron clypearia (Jack) IC Nielsen;
Mimosaceae), a popular traditional Chinese medicine, has a significant anti-inflammatory …

In Vitro and In Vivo Antipsoriatic Efficacy of Protected and Unprotected Sugar–Zinc Phthalocyanine Conjugates

S Makuch, P Kupczyk, M Woźniak, A Makarec… - Pharmaceutics, 2024 - mdpi.com
Psoriasis, a chronic immune-mediated skin disorder affecting over 125 million people
globally, is characterized by abnormal keratinocyte proliferation and immune cell infiltration …

[HTML][HTML] Dysregulated dermal mesenchymal stem cell proliferation and differentiation interfered by glucose metabolism in psoriasis

X Zhao, J Xing, J Li, R Hou, X Niu… - … Journal of Stem …, 2021 - synapse.koreamed.org
Methods and Results We found that the OCR of DMSCs in psoriatic lesions was higher than
that in the control group, and mRNA of GLUT1 and HK2 were up-regulated compared with …

[HTML][HTML] The impact of glucose conjugation on the activity and uptake of zinc phthalocyanine in HaCaT keratinocytes stimulated with proinflammatory cytokines

S Makuch, P Ziółkowski, M Woźniak - Photodiagnosis and Photodynamic …, 2024 - Elsevier
Significance Glucose metabolism has been proven as an essential process for proliferating
keratinocytes, which highlights the importance of glucose transporter-1 (GLUT1) not only in …

Developments in carbohydrate-based metzincin inhibitors

D Cuffaro, E Nuti, F D'Andrea, A Rossello - Pharmaceuticals, 2020 - mdpi.com
Matrix metalloproteinases (MMPs) and A disintegrin and Metalloproteinase (ADAMs) are
zinc-dependent endopeptidases belonging to the metzincin superfamily. Upregulation of …