Diversity-Orientated Synthesis and Biological Properties of Compounds Based on the N-Phenylquinoneimine Scaffold
The N-phenylquinoneimine scaffold is a versatile synthetic platform that has gained
significant attention in the field of drug discovery due to its structural diversity and capacity to …
significant attention in the field of drug discovery due to its structural diversity and capacity to …
Cu‐Catalyzed Chan–Evans–Lam Coupling Reactions of 2‐Nitroimidazole with Aryl Boronic Acids: An Effort toward New Bioactive Agents against S. pneumoniae
S Raju, PE Sheridan, AK Hauer… - Chemistry & …, 2022 - Wiley Online Library
The coupling of phenylboronic acids with poorly‐activated imidazoles is studied as a model
system to explore the use of copper‐catalyzed Chan–Evans–Lam (CEL) coupling for …
system to explore the use of copper‐catalyzed Chan–Evans–Lam (CEL) coupling for …
Cu−NHC Complex for Chan‐Evans‐Lam Cross‐Coupling Reactions of N‐Heterocyclic Compounds and Arylboronic Acids
An efficient copper (II) N‐heterocyclic carbene (NHC) complex with an NCN coordination
mode was optimized to catalyze the Chan–Evans‐Lam (CEL) cross‐coupling reaction of …
mode was optimized to catalyze the Chan–Evans‐Lam (CEL) cross‐coupling reaction of …
Exploiting Iminoquinones as Electrophilic at Nitrogen “N+” Synthons for C–N Bond Construction
LM Mori-Quiroz, CG Comadoll, JE Super… - Organic Letters, 2021 - ACS Publications
New methods for C–N bond construction exploiting the N-centered electrophilic character of
iminoquinones are reported. Iminoquinones, generated in situ via the condensation of o …
iminoquinones are reported. Iminoquinones, generated in situ via the condensation of o …
Cu‐Catalyzed Cross‐Coupling Reactions of Enamines and Terminal Alkynes: Access of Propargylamines as Neurodegenerative Disorder Agents
L Mohan, JE Lee, M Srinivasarao… - Asian Journal of …, 2023 - Wiley Online Library
Reactions between enamine analogues and terminal alkynes were explored. Copper (I)
complex of 1, 10‐phenanthroline catalyzed these reactions to generate a diastereoselective …
complex of 1, 10‐phenanthroline catalyzed these reactions to generate a diastereoselective …
Photocatalytic Annulation of Enaminones with Thioureas for the Synthesis of 2-Aminothiazoles via Tandem C–S and C–N Bond Formation
Q Huang, C Wan, JP Wan - Synthesis, 2024 - thieme-connect.com
Visible-light photocatalytic reactions between enaminones and thioureas leading to thiazole
products have been achieved. The annulation process consists of tandem C–S and C–N …
products have been achieved. The annulation process consists of tandem C–S and C–N …
Radical aminoalkylation of maleimides with alkylamines and alkanes
J Li, W Zhang, YA Li, G Wu… - Applied Organometallic …, 2023 - Wiley Online Library
A meaningful copper‐catalyzed chemo‐selective oxidative alkylamination of maleimides
with secondary alkyl amines and simple alkanes has been developed. This transformation …
with secondary alkyl amines and simple alkanes has been developed. This transformation …
Sodium Trifluoroacetate mediated Copper-Catalyzed aza-Michael addition of α, β-unsaturated olefins with aromatic amines
We present a sodium trifluoroacetate (CF 3 CO 2 Na) mediated copper-catalyzed aza-
Michael addition of aromatic amines with activated olefins under mild, aqueous reaction …
Michael addition of aromatic amines with activated olefins under mild, aqueous reaction …
Palladium-Catalyzed N-Alkenylation of N-Aryl Phosphoramidates with Alkenes
YA Li, G Wu, J Li - Molecules, 2023 - mdpi.com
Versatile and concise Pd-catalyzed oxidative N-alkenylation of N-aryl phosphoramidates
with alkenes is described in this study, a reaction that is of great significance but surprisingly …
with alkenes is described in this study, a reaction that is of great significance but surprisingly …
Synthetic approach to 2-alkyl-4-quinolones and 2-alkyl-4-quinolone-3-carboxamides based on common β-keto amide precursors
Y Mollova-Sapundzhieva, P Angelov… - Beilstein Journal of …, 2023 - beilstein-journals.org
Abstract β-Keto amides were used as convenient precursors to both 2-alkyl-4-quinolones
and 2-alkyl-4-quinolone-3-carboxamides. The utility of this approach is demonstrated with …
and 2-alkyl-4-quinolone-3-carboxamides. The utility of this approach is demonstrated with …