Amorphous solid dispersions: Rational selection of a manufacturing process

T Vasconcelos, S Marques, J das Neves… - Advanced drug delivery …, 2016 - Elsevier
Amorphous products and particularly amorphous solid dispersions are currently one of the
most exciting areas in the pharmaceutical field. This approach presents huge potential and …

A systematic and robust assessment of hot-melt extrusion-based amorphous solid dispersions: Theoretical prediction to practical implementation

A Alzahrani, D Nyavanandi, P Mandati… - International Journal of …, 2022 - Elsevier
Amorphous solid dispersions (ASDs) have gained attention as a formulation strategy in
recent years, with the potential to improve the apparent solubility and, hence, the oral …

Coupling 3D printing with hot-melt extrusion to produce controlled-release tablets

J Zhang, X Feng, H Patil, RV Tiwari… - International journal of …, 2017 - Elsevier
The main objective of this work was to explore the potential of coupling fused deposition
modeling in three-dimensional (3D) printing with hot-melt extrusion (HME) technology to …

Hydroxypropyl methylcellulose-based controlled release dosage by melt extrusion and 3D printing: Structure and drug release correlation

J Zhang, W Yang, AQ Vo, X Feng, X Ye, DW Kim… - Carbohydrate …, 2017 - Elsevier
The objective of this study was to develop a new approach for fabrication of zero order
release of active pharmaceutical ingredients (APIs) using hot-melt extrusion (HME) and 3D …

Characterization of amorphous solid dispersions: An update

X Ma, RO Williams III - Journal of Drug Delivery Science and Technology, 2019 - Elsevier
Amorphous solid dispersions (ASDs) are a promising formulation approach to improve the
solubility, dissolution rate, and bioavailability of poorly water-soluble drugs. ASDs have …

Development of 3D printed tablets by fused deposition modeling using polyvinyl alcohol as polymeric matrix for rapid drug release

C Wei, NG Solanki, JM Vasoya, AV Shah… - Journal of …, 2020 - Elsevier
In this study, the processability of polyvinyl alcohol (PVA), a water-soluble polymer, into melt-
extruded filaments and then into 3D printed tablets by fused deposition modeling was …

Development and evaluation of an oral fast disintegrating anti-allergic film using hot-melt extrusion technology

MB Pimparade, A Vo, AS Maurya, J Bae… - European Journal of …, 2017 - Elsevier
The main objective of this novel study was to develop chlorpheniramine maleate orally
disintegrating films (ODF) using hot-melt extrusion technology and evaluate the …

Characterization of amorphous solid dispersions

X Liu, X Feng, RO Williams, F Zhang - Journal of Pharmaceutical …, 2018 - Springer
The study of amorphous solid dispersions (ASDs) is currently one of the most exciting areas
in pharmaceutics. Research has shown that ASDs offer unique advantages in improving the …

Application and limitations of thermogravimetric analysis to delineate the hot melt extrusion chemical stability processing window

DE Moseson, MA Jordan, DD Shah, ID Corum… - International Journal of …, 2020 - Elsevier
Thermogravimetric analysis (TGA) is frequently used to define the threshold of acceptable
processing temperatures for hot melt extrusion. Herein, evaluation of chemical stability of …

Polymer–surfactant system based amorphous solid dispersion: Precipitation inhibition and bioavailability enhancement of itraconazole

D Feng, T Peng, Z Huang, V Singh, Y Shi, T Wen, M Lu… - Pharmaceutics, 2018 - mdpi.com
The rapid release of poorly water-soluble drugs from amorphous solid dispersion (ASD) is
often associated with the generation of supersaturated solution, which provides a strong …