Heterocycles are an extraordinarily important class of compounds, making up more than half
of all known organic compounds. Heterocycles are present in a wide variety of drugs, most …

The oxazole is a five-membered aromatic heterocycle that contains both oxygen and
nitrogen. Oxazoles are numbered around the ring starting at the oxygen atom as shown …

Synthesis of Functionalized Oxazolines and Oxazoles with DAST and Deoxo-Fluor |
Organic Letters ACS ACS Publications C&EN CAS Find my institution Log In Organic …

Cyanobacteria from a diversity of marine and freshwater habitats are known to produce
neurotoxic secondary metabolites. 1 Herein, we describe the complete stereostructure …

We have achieved a total synthesis of telomestatin, and its absolute configuration was
determined to be (R). Coupling of cysteine-containing trisoxazole amine and serine …

A novel total synthesis of apratoxin A is described, with key steps including the assembly of
its ketide segment through ad‐proline‐catalyzed direct aldol reaction and Oppolzer's anti …

The isolation of the cytotoxic Lissoclinum sp. metabolite trunkamide A was reported in 1996.
After completion of a total synthesis in 1999, it became clear that the structure of this marine …

New methodology for the synthesis of variously substituted 2-oxazolines and one
dihydrooxazine using aldehydes, amino alcohols, and N-bromosuccinimide as an oxidizing …

A new class of tridentate bis (oxazoline) ligands 7, in which an N-phenylaniline unit links the
two oxazoline rings, has been prepared. The key step in their synthesis is a Hartwig …

An expedient method for the direct conversion of aldehydes to 2, 4-disubstituted oxazoles is
presented. The method relies on the oxidation of an oxazolidine formed from the …