Discovery of sulfadrug–pyrrole conjugates as carbonic anhydrase and acetylcholinesterase inhibitors
Human carbonic anhydrase (hCA) isoenzymes are zinc ion‐containing, widespread
metalloenzymes and they classically play a role in pH homeostasis maintenance. CA …
metalloenzymes and they classically play a role in pH homeostasis maintenance. CA …
Determination of Antioxidant, Anti-Alzheimer, Antidiabetic, Antiglaucoma and Antimicrobial Effects of Zivzik Pomegranate (Punica granatum)—A Chemical Profiling by …
H Karagecili, E İzol, E Kirecci, İ Gulcin - Life, 2023 - mdpi.com
Zivzik pomegranate (Punica granatum) has recently sparked considerable interest due to its
nutritional and antioxidant properties. To evaluate the antioxidant capacities of P. granatum …
nutritional and antioxidant properties. To evaluate the antioxidant capacities of P. granatum …
[HTML][HTML] Synthesis and inhibition profiles of N-benzyl-and N-allyl aniline derivatives against carbonic anhydrase and acetylcholinesterase–A molecular docking study
The alkyl and aryl derivatives of aniline are important starting materials in fine organic
synthesis. Allyl bromide and benzyl chloride were taken as substrates for the alkylation …
synthesis. Allyl bromide and benzyl chloride were taken as substrates for the alkylation …
Comprehensive Metabolite Profiling of Cinnamon (Cinnamomum zeylanicum) Leaf Oil Using LC-HR/MS, GC/MS, and GC-FID: Determination of Antiglaucoma …
In this study, for the first time, the antioxidant and antidiabetic properties of the essential oil
from cinnamon (Cinnamomum zeylanicum) leaves were evaluated and investigated using …
from cinnamon (Cinnamomum zeylanicum) leaves were evaluated and investigated using …
Evaluation of the in vitro antioxidant, antidiabetic and anticholinergic properties of rosmarinic acid from rosemary (Rosmarinus officinalis L.)
M Topal, İ Gulcin - Biocatalysis and Agricultural Biotechnology, 2022 - Elsevier
In this study, antidiabetic, anticholinergic, and antioxidant abilities of rosmarinic acid were
evaluated and compared to standards. To determine its antioxidant activity different in vitro …
evaluated and compared to standards. To determine its antioxidant activity different in vitro …
Antioxidant, antidiabetic, anticholinergic, and antiglaucoma effects of magnofluorine
Magnofluorine, a secondary metabolite commonly found in various plants, has
pharmacological potential; however, its antioxidant and enzyme inhibition effects have not …
pharmacological potential; however, its antioxidant and enzyme inhibition effects have not …
Screening of carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase, and α-glycosidase enzyme inhibition effects and antioxidant activity of coumestrol
Coumestrol (3, 9-dihydroxy-6-benzofuran [3, 2-c] chromenone) as a phytoestrogen and
polyphenolic compound is a member of the Coumestans family and is quite common in …
polyphenolic compound is a member of the Coumestans family and is quite common in …
Isofraxidin: Antioxidant, Anti‐carbonic Anhydrase, Anti‐cholinesterase, Anti‐diabetic, and in Silico Properties
The development of innovative pharmacological formulations for the treatment and
prevention of various major diseases, including cancer, diabetes, and glaucoma, has been …
prevention of various major diseases, including cancer, diabetes, and glaucoma, has been …
Synthesis and Evaluation of Quinazolin‐4(3H)‐one Derivatives as Multitarget Metabolic Enzyme Inhibitors: A Biochemistry‐Oriented Drug Design
In this study, imines bearing quinazolin‐4 (3H)‐one were synthesized and their inhibitory
properties were investigated against some metabolic enzymes including …
properties were investigated against some metabolic enzymes including …
Synthesis of new carboxylates and sulfonates containing thiazolidin-4-one ring and evaluation of inhibitory properties against some metabolic enzymes
A series of thizaolidin-4-one derivatives (3a-o) was synthesized with excellent yield (94–
97%) and the structures of the compounds were characterized with Fourier-transform …
97%) and the structures of the compounds were characterized with Fourier-transform …