Role of sulphur-heterocycles in medicinal chemistry: An update
From many decades, S-heterocycles have maintained their status as an important part and
core of FDA approved drugs and medicinally active compounds. With exhaustive exploration …
core of FDA approved drugs and medicinally active compounds. With exhaustive exploration …
A decade update on the application of β-oxodithioesters in heterocyclic synthesis
ZB Dong, Z Gong, Q Dou, B Cheng… - Organic & Biomolecular …, 2023 - pubs.rsc.org
The diversified synthesis of heterocyclic compounds has always been one of the popular
subjects of organic chemistry. To this end, great efforts have been devoted to developing …
subjects of organic chemistry. To this end, great efforts have been devoted to developing …
Base-Promoted Reaction of 4-Chloro-3-vinyl Coumarins, Phenacylpyridinium Bromides, and Elemental Sulfur: A Designed Approach to Thiopyrano [4, 3-c] chromen-5 …
B Farajpour, A Alizadeh - The Journal of Organic Chemistry, 2022 - ACS Publications
A designed synthesis of thiopyrano [4, 3-c] chromen-5 (1 H)-ones was developed based on
a base-promoted three-component reaction between 4-chloro-3-vinyl coumarins …
a base-promoted three-component reaction between 4-chloro-3-vinyl coumarins …
Regio- and Chemoselective Access to Dihydrothiophenes and Thiophenes via Halogenation/Intramolecular C(sp2)–H Thienation of α-Allyl Dithioesters at Room …
G Shukla, K Raghuvanshi… - The Journal of Organic …, 2022 - ACS Publications
An operationally simple, practical, and efficient cascade approach employing α-allyl
dithioesters and NBS/NIS has been achieved to access a series of dihydrothiophenes and …
dithioesters and NBS/NIS has been achieved to access a series of dihydrothiophenes and …
Assembly of fully substituted 2, 5-dihydrothiophenes via a novel sequential multicomponent reaction
A new and efficient synthesis of fully substituted 2, 5-dihydrothiophenes by a sequential one-
pot four component reaction between primary amines, β-ketoesters, aryl isothiocyanates and …
pot four component reaction between primary amines, β-ketoesters, aryl isothiocyanates and …
Regioselective synthesis of dihydrothiophenes and thiophenes via the rhodium-catalyzed transannulation of 1, 2, 3-thiadiazoles with alkenes
JY Son, J Kim, SH Han, SH Kim, PH Lee - Organic letters, 2016 - ACS Publications
A method for the regioselective synthesis of a wide range of dihydrothiophenes was
developed from the rhodium-catalyzed transannulation of 1, 2, 3-thiadiazoles with aliphatic …
developed from the rhodium-catalyzed transannulation of 1, 2, 3-thiadiazoles with aliphatic …
Access to Fully Substituted Thiazoles and 2,3-Dihydrothiazoles via Copper-Catalyzed [4 + 1] Heterocyclization of α-(N-Hydroxy/aryl)imino-β-oxodithioesters with α …
An efficient chemoselective practical route to fully substituted thiazoles and 2, 3-
dihydrothiazoles has been devised by [4+ 1] heterocyclization of α-(N-hydroxy/aryl) imino-β …
dihydrothiazoles has been devised by [4+ 1] heterocyclization of α-(N-hydroxy/aryl) imino-β …
p-TSA/Base-Promoted Propargylation/Cyclization of β-Ketothioamides for the Regioselective Synthesis of Highly Substituted (Hydro)thiophenes
Metal-free, p-toluenesulfonic acid (p-TSA)-mediated, straightforward propargylation of β-
ketothioamides with aryl propargyl alcohol has been achieved at room temperature. In …
ketothioamides with aryl propargyl alcohol has been achieved at room temperature. In …
Metal-free one-pot four-component cascade annulation in ionic liquids at room temperature: convergent access to Thiazoloquinolinone derivatives
A Singh, A Srivastava, MS Singh - The Journal of Organic …, 2018 - ACS Publications
An efficient, eco-friendly, and highly convergent one-pot route to privileged
thiazoloquinolinone derivatives has been developed via four-component cascade coupling …
thiazoloquinolinone derivatives has been developed via four-component cascade coupling …
Copper-catalyzed one-pot cross-dehydrogenative thienannulation: Chemoselective access to naphtho [2, 1-b] thiophene-4, 5-diones and subsequent transformation …
A facile, cost-effective, and highly efficient copper-catalyzed, TEMPO-mediated
straightforward synthesis of 2, 3-disubstituted naphtho [2, 1-b] thiophene-4, 5-diones has …
straightforward synthesis of 2, 3-disubstituted naphtho [2, 1-b] thiophene-4, 5-diones has …