Radiometallation and photo-triggered release of ready-to-inject radiopharmaceuticals from the solid phase
D Śmiłowicz, S Eisenberg, SH Ahn, AJ Koller… - Chemical …, 2023 - pubs.rsc.org
The efficient, large-scale synthesis of radiometallated radiopharmaceuticals represents an
emerging clinical need which, to date, is inherently limited by time consuming, sequential …
emerging clinical need which, to date, is inherently limited by time consuming, sequential …
A UV-Vis method for investigation of gallium (iii) complexation kinetics with NOTA and TRAP chelators: Advantages, limitations and comparison with radiolabelling
V Lebruška, T Dobrovolná, T Gemperle… - Dalton …, 2024 - pubs.rsc.org
An easy and cheap method for measurement of GaIII complexation kinetics was developed.
The method is based on UV-Vis quantification of non-complexed chelators after the addition …
The method is based on UV-Vis quantification of non-complexed chelators after the addition …
Expedient Access to 18F‐Fluoroheteroarenes via Deaminative Radiofluorination of Aniline‐Derived Pyridinium Salts
J Ford, S Ortalli, Z Chen, JBI Sap… - Angewandte …, 2024 - Wiley Online Library
Herein, we disclose that pyridinium salts derived from abundant (hetero) anilines represent
a novel precursor class for nucleophilic aromatic substitution reactions with [18F] fluoride …
a novel precursor class for nucleophilic aromatic substitution reactions with [18F] fluoride …
(Radio) Fluorination Reactions for the Synthesis of Aryl Fluorides: Recent Advances and Perspectives
J Han, ZM Zhang - European Journal of Organic Chemistry, 2024 - Wiley Online Library
The formation of carbon‐fluorine (C− F) bonds is an important research field in organic
synthesis because inserting a fluorine atom into an organic compound can alter its …
synthesis because inserting a fluorine atom into an organic compound can alter its …
Transition-Metal-Mediated Radiohalogenation using Aryl Boron Reagents
VK Burianova, H McErlain, A Sutherland - Synthesis, 2024 - thieme-connect.com
Biomolecules labeled with radioisotopes of iodine and fluorine play a major role in science
and medicine, with a range of applications including molecular imaging of disease, as …
and medicine, with a range of applications including molecular imaging of disease, as …
Fluorine-18 or Gallium-68: The Perspective of PET Radiochemist
RN Krasikova - Radiochemistry, 2023 - Springer
Abstract Two radionuclides, 18F (T 1/2 110 min) and 68Ga (T 1/2 68 min), currently play the
leading role in the development of positron emission tomography (PET). This review …
leading role in the development of positron emission tomography (PET). This review …
GMP-Compliant Automated Radiolabeling and Quality Controls of [68Ga] Ga-FAPI-46 for Fibroblast Activation Protein-Targeted PET Imaging in Clinical Settings
L Rubira, J Torchio, J Fouillet, J Vanney… - Chemical and …, 2024 - jstage.jst.go.jp
In nuclear medicine, molecular imaging of the tumor microenvironment using
radiopharmaceuticals (RPs) targeting cancer-associated fibroblasts is gaining significant …
radiopharmaceuticals (RPs) targeting cancer-associated fibroblasts is gaining significant …
Ftor-18 ili Galliy-68: mnenie PET radiokhimika
RN Krasikova - Radiohimiâ, 2023 - journals.rcsi.science
На данном этапе развития позитронной эмиссионной томографии (ПЭТ) лидирующую
роль играют два радионуцлида-18 F (T 1/2 110 мин) и 68 Ga (T 1/2 68 мин). В …
роль играют два радионуцлида-18 F (T 1/2 110 мин) и 68 Ga (T 1/2 68 мин). В …