The 1, 2-diamine moiety is an ubiquitous structural motif found in a wealth of natural
products, including non-proteinogenic amino acids and alkaloids, in pharmaceutical agents …

We report the use of electrochemistry to perform a direct oxidative dearomatization of
indoles leading to 2, 3-dialkoxy or 2, 3-diazido indolines under undivided conditions at a …

As the aromatic tryptophan (Trp) side chain plays a pivotal role in influencing the structure
and function of peptides and proteins, it has become an attractive target for the late‐stage …

This Account summarizes our involvement in the development of dearomatization reactions
of indoles that has for origin a total synthesis problematic. We present the effort from our …

1, 3-Dipolar cycloaddition of organic azides 1, 2, or 3 to acetylenic amides 4 or 5 under
solvent-free microwave irradiation produced the corresponding N-substituted C-carbamoyl …

Tetrahedron Letters,Vo1.27,No.25,pp 2809-2812‘1986 0040-4039/86 $3.00 + .OO Printed in
Great Britain Pergamon Journals Ltd. A Page 1 Tetrahedron Letters,Vo1.27,No.25,pp …

Efficient copper-catalyzed aerobic oxidative dearomatization of indoles with trimethylsilyl
azide (TMSN3) for the synthesis of 2-azidoindolin-3-ols has been developed. Molecular …

Use of 3-azidoindoles in organic synthesis remains a difficult task owing to their instabilities.
Herein, we report a general and concise approach for tackling this problem by using 3 …

Triazole-oligomers by 1,3-dipolar cycloaddition Page 1 Issue in Honor of Prof. Edmunds
Lukevics ARKIVOC 2006 (v) 43-62 ISSN 1424-6376 Page 43 © ARKAT Triazole-oligomers …

Reactions of 3-lithiopropiolate 10 with isocyanates or diisocyanates gave
monocarbamoylpropiolates 11a, b and bis-carbamoylpropiolates 12a-d, in 40-76% yields. 1 …